| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA804767 | B | Inhibitory activity of compound against SSAT extracted from superinduced H157 cells | 2 | ALA1134460 | cell-based format | Scientific Literature | ||
| 2. | ALA872601 | B | Inhibitory activity against human SSAT | 1 | ALA1134460 | single protein format | Scientific Literature | ||
| 3. | ALA804768 | B | Effect of 10 uM on spermine/spermidine-N-acetyltransferase (SSAT) induction in non-SCLC cells | 18 | ALA1134460 | cell-based format | Scientific Literature | ||
| 4. | ALA955109 | B | Inhibition of spermidine/spermine N1-acetyltransferase activity in human SK-MEL cells at 10 uM after 24 hrs relative to control | Homo sapiens | 3 | ALA1153376 | cell-based format | Scientific Literature | |
| 5. | ALA2185110 | B | Activity of SSAT in human DU145 cells assessed per ug DNA at 100 uM after 72 hrs in presence of serum amine oxidase inhibitor aminoguanidine (RVb = 62 +/- 4 pmol/h per ug DNA) | Homo sapiens | 4 | ALA2177009 | cell-based format | Scientific Literature | |
| 6. | ALA2185111 | B | Activity of SSAT in human DU145 cells assessed per ug DNA at 100 uM after 48 hrs in presence of serum amine oxidase inhibitor aminoguanidine (RVb = 58 pmol/h per ug DNA) | Homo sapiens | 4 | ALA2177009 | cell-based format | Scientific Literature | |
| 7. | ALA2185112 | B | Activity of SSAT in human DU145 cells assessed per ug DNA at 100 uM after 24 hrs in presence of serum amine oxidase inhibitor aminoguanidine (RVb = 59 +/- 1 pmol/h per ug DNA) | Homo sapiens | 4 | ALA2177009 | cell-based format | Scientific Literature | |
| 8. | ALA3242686 | B | Inhibition of human SSAT using spermidine as substrate | Homo sapiens | 2 | ALA3232957 | single protein format | Scientific Literature | |
| 9. | ALA3538524 | A | Drug level in human HepG2 cells assessed as SSAT1-mediated compound formation treated with SpmTrien at 100 uM for 24 hrs pretreated with 50 uM DENSpm for 24 hrs | Homo sapiens | 2 | ALA3526099 | cell-based format | Scientific Literature | |
| 10. | ALA3538525 | A | Drug metabolism in human HepG2 cells assessed as SSAT1-mediated (N12-acetyl)-1,12-diamino-3,6,9-triazadodecane formation at 100 uM for 24 hrs pretreated with 50 uM DENSpm for 24 hrs | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 11. | ALA3538795 | A | Drug metabolism in human HepG2 cells assessed as SSAT1-mediated (N1-acetyl)-1,12-diamino-3,6,9-triazadodecane formation at 100 uM for 24 hrs in presence of SSAT2 shRNA | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 12. | ALA3538796 | A | Drug level in human HepG2 cells assessed as SSAT1-mediated compound formation treated with SpmTrien at 100 uM for 24 hrs in presence of SSAT2 shRNA | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 13. | ALA3541423 | A | Activity of human recombinant SSAT1 | Homo sapiens | 1 | ALA3526099 | single protein format | Scientific Literature | |
| 14. | ALA3541424 | A | Activity of human recombinant SSAT1 assessed as compound formation treated with 1 mM SpmTrien for 50 mins by HPLC analysis | Homo sapiens | 2 | ALA3526099 | single protein format | Scientific Literature | |
| 15. | ALA3541431 | A | Drug metabolism in human HepG2 cells assessed as SSAT1-mediated (N1-acetyl)-spermidine formation at 100 uM for 24 hrs | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 16. | ALA3541432 | A | Drug metabolism in human HepG2 cells assessed as SSAT1-mediated (N1-acetyl)-spermine formation at 100 uM for 24 hrs | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 17. | ALA3541434 | A | Drug level in human HepG2 cells assessed as SSAT1-mediated compound formation treated with SpmTrien at 100 uM for 24 hrs | Homo sapiens | 3 | ALA3526099 | cell-based format | Scientific Literature | |
| 18. | ALA3541436 | A | Drug metabolism in human HepG2 cells assessed as SSAT1-mediated (N1-acetyl)-1,12-diamino-3,6,9-triazadodecane formation at 100 uM for 24 hrs | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 19. | ALA3541439 | A | Drug level in human HepG2 cells assessed as SSAT1-mediated compound formation per ug DNA treated with Spm Trien at 100 uM for 24 hrs | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature | |
| 20. | ALA3541442 | A | Drug metabolism in human HepG2 cells assessed as SSAT1-mediated (N1-acetyl)-1,12-diamino-3,6,9-triazadodecane formation at 100 uM for 24 hrs pretreated with 50 uM DENSpm for 24 hrs | Homo sapiens | 1 | ALA3526099 | cell-based format | Scientific Literature |
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