# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3378282 | B | Inhibition of PDHK3 (unknown origin) | Homo sapiens | 1 | ALA3352550 | single protein format | Scientific Literature | |
2. | ALA3378295 | B | Inhibition of recombinant PDHK3 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISA | Homo sapiens | 1 | ALA3352550 | assay format | Scientific Literature | |
3. | ALA3998679 | B | Inhibition of recombinant human PDK3 in presence of E1 protein incubated for 10 mins by titration assay | Homo sapiens | 1 | ALA3997786 | single protein format | Scientific Literature | |
4. | ALA3998683 | B | Inhibition of recombinant human PDK3 in presence of E1 protein and PDC core E2/E3BP incubated for 10 mins by titration assay | Homo sapiens | 1 | ALA3997786 | single protein format | Scientific Literature | |
5. | ALA4008868 | B | Inhibition of fluorescein-labelled VER160364 binding to PDHK3 (unknown origin) after 90 mins by fluorescence polarization assay | Homo sapiens | 1 | ALA4007418 | single protein format | Scientific Literature | |
6. | ALA4008878 | B | Inhibition of PDHK3 (unknown origin) assessed as decrease in phosphorylation of E1alpha subunit at serine 293 residue after 1 hr by DELFIA | Homo sapiens | 2 | ALA4007418 | single protein format | Scientific Literature | |
7. | ALA4009662 | B | Inhibition of PDK3 (unknown origin) using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 4 | ALA4007440 | single protein format | Scientific Literature | |
8. | ALA4009663 | B | Inhibition of PDK3 (unknown origin) assessed as inactivation rate using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
9. | ALA4009664 | B | Ratio of Kinact to Ki for PDK3 (unknown origin) | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
10. | ALA4311230 | B | Binding affinity to SUMO-fused/His-tagged PDK3 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysis | Homo sapiens | 4 | ALA4308888 | assay format | Scientific Literature | |
11. | ALA4366665 | B | Inhibition of human PDK3 at 100 nM using MBP as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
12. | ALA4369504 | B | Inhibition of PDK3 (unknown origin) using PDC E1 as substrate measured after 30 mins by kinase-glo assay | Homo sapiens | 4 | ALA4368877 | single protein format | Scientific Literature | |
13. | ALA4400361 | B | Inhibition of PDK3 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assay | Homo sapiens | 1 | ALA4396967 | single protein format | Scientific Literature | |
14. | ALA4403264 | B | Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assay | Homo sapiens | 24 | ALA4402524 | single protein format | Scientific Literature | |
15. | ALA4403270 | B | Inhibition of PDHK3 (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4402524 | single protein format | Scientific Literature | |
16. | ALA4405629 | B | Inhibition of PDHK3 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4402587 | single protein format | Scientific Literature | |
17. | ALA4413205 | B | Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminescence assay | Homo sapiens | 4 | ALA4411306 | assay format | Scientific Literature | |
18. | ALA4737392 | B | Binding affinity to PDK3 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA4732185 | single protein format | Scientific Literature | |
19. | ALA4824990 | B | Inhibition of human PDHK3 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrate preincubated with enzyme complex for 45 mins followed by ATP addition and then later incubated with substrate for 90 mins by absorption spectrophotometric assay | Homo sapiens | 1 | ALA4823293 | single protein format | Scientific Literature |