| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1001232 | B | Inhibition of PDHK4 | 1 | single protein format | Scientific Literature | |||
| 2. | ALA1116751 | B | Inhibition of PDHK4 at 5 uM | 1 | single protein format | Scientific Literature | |||
| 3. | ALA1959341 | B | Inhibition of human His-tagged PDHK4 using biotin-YHGHSMSDPGVSYRRR-amide as substrate after 20 mins by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA2015474 | B | Inhibition of PDHK4 at 10 uM | 1 | single protein format | Scientific Literature | |||
| 5. | ALA3378296 | B | Inhibition of recombinant PDHK4 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISA | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA3998680 | B | Inhibition of recombinant human PDK4 in presence of E1 protein incubated for 10 mins by titration assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA3998684 | B | Inhibition of recombinant human PDK4 in presence of E1 protein and PDC core E2/E3BP incubated for 10 mins by titration assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4008869 | B | Inhibition of fluorescein-labelled VER160364 binding to PDHK4 (unknown origin) after 90 mins by fluorescence polarization assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4008879 | B | Inhibition of PDHK4 (unknown origin) assessed as decrease in phosphorylation of E1alpha subunit at serine 293 residue after 1 hr by DELFIA | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 10. | ALA4009666 | B | Inhibition of PDK4 (unknown origin) at 10 uM using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 11. | ALA4009667 | B | Inhibition of PDK4 (unknown origin) using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4191103 | B | Inhibition of recombinant full-length human PDHK4 at 1 uM using KKKYHGHSMSDPGVSYRT as substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4311231 | B | Binding affinity to SUMO-fused/His-tagged PDK4 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysis | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 14. | ALA4314905 | B | Inhibition of recombinant full-length human PDHK4 assessed as residual activity at 10 uM using KKKYHGHSMSDPGVSYRT as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA4333047 | B | Inhibition of PDK4 (unknown origin) at 1 uM relative to control | Homo sapiens | 24 | single protein format | Scientific Literature | ||
| 16. | ALA4333048 | B | Inhibition of PDK4 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 17. | ALA4333049 | B | Inhibition of PDK4 in HEK293T cells assessed as reduction in PDHE1alpha phosphorylation at Ser-232 residue by measuring phosphorylated PDHE1alpha level at 10 uM after 24 hrs by Western blot analysis (Rvb = 1 No_unit) | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA4333050 | B | Inhibition of PDK4 in HEK293T cells assessed as reduction in PDHE1alpha phosphorylation at Ser-293 residue by measuring phosphorylated PDHE1alpha level at 10 uM after 24 hrs by Western blot analysis (Rvb = 1 No_unit) | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 19. | ALA4333051 | B | Inhibition of PDK4 in HEK293T cells assessed as reduction in PDHE1alpha phosphorylation at Ser-300 residue by measuring phosphorylated PDHE1alpha level at 10 uM after 24 hrs by Western blot analysis (Rvb = 1 No_unit) | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 20. | ALA4333052 | B | Inhibition of PDK4 in HEK293T cells assessed as reduction in PDHE1alpha phosphorylation at Ser-232 residue by measuring phosphorylated PDHE1alpha level at 5 mM after 24 hrs by Western blot analysis (Rvb = 1 No_unit) | Homo sapiens | 1 | cell-based format | Scientific Literature |
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