| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA858390 | B | Apparent binding constant for purified human kidney TPMT | Homo sapiens | 14 | ALA1123412 | tissue-based format | Scientific Literature | |
| 2. | ALA814140 | B | Inhibition of purified human kidney thiopurine methyltransferase (TPMT) | 27 | ALA1123412 | single protein format | Scientific Literature | ||
| 3. | ALA3369580 | B | Binding affinity to thiopurine methyltransferase (unknown origin) by NMR analysis | Homo sapiens | 1 | ALA3351755 | single protein format | Scientific Literature | |
| 4. | ALA4416334 | A | Inhibition of human TPMT expressed in Escherichia coli assessed as reduction in SAH level at 10 uM using 6-mercaptopurine as substrate in presence of SAM incubated for 30 mins by LC-MS/MS analysis relative to control | Homo sapiens | 1 | ALA4414609 | assay format | Scientific Literature | |
| 5. | ALA4416341 | A | Inhibition of human TPMT expressed in Escherichia coli assessed as reduction in SAH level at 1 uM using 6-mercaptopurine as substrate in presence of SAM incubated for 30 mins by LC-MS/MS analysis relative to control | Homo sapiens | 1 | ALA4414609 | assay format | Scientific Literature | |
| 6. | ALA4416355 | A | Inhibition of human TPMT expressed in Escherichia coli assessed as reduction in SAH level using 6-mercaptopurine as substrate in presence of SAM incubated for 30 mins by LC-MS/MS analysis | Homo sapiens | 1 | ALA4414609 | assay format | Scientific Literature |
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