# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA679630 | B | Compound was tested for inhibition against estrogen sulfotransferase (EST), a human cytosolic sulfotransferase | 1 | ALA1135027 | single protein format | Scientific Literature | ||
2. | ALA679631 | B | Compound was tested for inhibition against estrogen sulfotransferase (EST), a human cytosolic sulfotransferase. | 1 | ALA1135027 | single protein format | Scientific Literature | ||
3. | ALA873654 | B | Inhibitory activity of compound was determined against estrogen sulfotransferase at 100 uM | 1 | ALA1135027 | single protein format | Scientific Literature | ||
4. | ALA682287 | B | Inhibitory activity of compound was determined against human estrogen sulfotransferase at 100 uM | 1 | ALA1135027 | single protein format | Scientific Literature | ||
5. | ALA909428 | B | Inhibition of human estrogen sulfotransferase | Homo sapiens | 9 | ALA1137329 | single protein format | Scientific Literature | |
6. | ALA1743309 | A | Major substrate of human cytosolic sulfotransferase SULT1E1 | Homo sapiens | 15 | ALA1743201 | single protein format | Scientific Literature | |
7. | ALA3540602 | A | Activity of human SULT1E1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | ALA3525912 | assay format | Scientific Literature | |
8. | ALA3540605 | A | Activity of human SULT1E1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | ALA3525912 | assay format | Scientific Literature | |
9. | ALA3539756 | A | Drug metabolism assessed as human SULT1E1-mediated (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[1,2-f][1,2,4]triazin-6-yloxy)propane-2-sulfonic acid formation at 2 and 20 uM for 30 mins by LC/MS analysis in presence of PAPS | Homo sapiens | 1 | ALA3526086 | single protein format | Scientific Literature | |
10. | ALA3540072 | A | Activity of human SULT1E1 assessed as compound formation treated with 2 and 20 uM brivanib for 30 mins by LC/MS analysis in presence of PAPS | Homo sapiens | 1 | ALA3526086 | single protein format | Scientific Literature | |
11. | ALA3537877 | A | Activity of SULT1E1 (unknown origin) | Homo sapiens | 1 | ALA3525919 | single protein format | Scientific Literature | |
12. | ALA4482695 | B | Substrate activity at SULT1E1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Km incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | ALA4482315 | cell-based format | Patent Bioactivity Data | |
13. | ALA4482696 | B | Substrate activity at SULT1E1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | ALA4482315 | cell-based format | Patent Bioactivity Data | |
14. | ALA4482697 | B | Substrate activity at SULT1E1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax/Km ratio level incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | ALA4482315 | cell-based format | Patent Bioactivity Data | |
15. | ALA4482698 | B | Substrate activity at SULT1A3 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Km incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | ALA4482315 | cell-based format | Patent Bioactivity Data | |
16. | ALA4482699 | B | Substrate activity at SULT1A3 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | ALA4482315 | cell-based format | Patent Bioactivity Data | |
17. | ALA4482700 | B | Substrate activity at SULT1A3 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax/Km ratio incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | ALA4482315 | cell-based format | Patent Bioactivity Data | |
18. | ALA4701345 | B | Inhibition of estrogen sulfotransferase in human liver cytosol incubated for 30 mins in presence of [3H]-estradiol and adenosine -3'-phosphate 5'-phosphosulfate by liquid scintillation counting method | Homo sapiens | 1 | ALA4699466 | subcellular format | Scientific Literature |