| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA666249 | A | Inhibitory effect in formation of metabolic intermediate complex between Cytochrome P450 and racemic compound 2 initially, on pre-incubation with Racemic 2 (300 uM) at 30 uM | Oryctolagus cuniculus | 1 | ALA1121797 | single protein format | Scientific Literature | |
| 2. | ALA1167168 | A | Inhibition of human recombinant CYP3A5 at 10 uM by spectrofluorimetry | Homo sapiens | 3 | ALA1165972 | single protein format | Scientific Literature | |
| 3. | ALA1658787 | A | Activity of human recombinant CYP3A5 assessed as compound remaining | Homo sapiens | 1 | ALA1649403 | single protein format | Scientific Literature | |
| 4. | ALA1743482 | A | Mechanism based inhibition of human cytochrome P450 3A5 | Homo sapiens | 1 | ALA1743341 | single protein format | Scientific Literature | |
| 5. | ALA1743483 | A | Mechanism based inhibition of human cytochrome P450 3A5 | Homo sapiens | 3 | ALA1743341 | single protein format | Scientific Literature | |
| 6. | ALA1743484 | A | Mechanism based inhibition of human cytochrome P450 3A5 | Homo sapiens | 1 | ALA1743341 | single protein format | Scientific Literature | |
| 7. | ALA1743485 | A | Mechanism based inhibition of human cytochrome P450 3A5 measured by testosterone hydroxylation | Homo sapiens | 2 | ALA1743341 | single protein format | Scientific Literature | |
| 8. | ALA1743486 | A | Mechanism based inhibition of human cytochrome P450 3A5 using expressed CYP3A5 cDNA | Homo sapiens | 1 | ALA1743341 | single protein format | Scientific Literature | |
| 9. | ALA1743513 | A | Mechanism based inhibition of human cytochrome P450 3A5, partition ratio | Homo sapiens | 1 | ALA1743341 | single protein format | Scientific Literature | |
| 10. | ALA1953082 | A | Inhibition of recombinant human CYP3A5 in supersomes using midazolam as substrate after 5 mins by LC-MS/MS analysis | Homo sapiens | 23 | ALA1949669 | single protein format | Scientific Literature | |
| 11. | ALA1953084 | A | Inhibition of recombinant human CYP3A5 in supersomes using midazolam as substrate at 60 uM after 5 mins by LC-MS/MS analysis | Homo sapiens | 17 | ALA1949669 | single protein format | Scientific Literature | |
| 12. | ALA1953085 | A | Inhibition of recombinant human CYP3A5 in supersomes using midazolam as substrate at 2 uM after 5 mins by LC-MS/MS analysis | Homo sapiens | 1 | ALA1949669 | single protein format | Scientific Literature | |
| 13. | ALA1960690 | A | Inhibition of CYP3A5 in human microsome | Homo sapiens | 1 | ALA1955765 | assay format | Scientific Literature | |
| 14. | ALA2044478 | A | Inhibition of CYP3A5 | 1 | ALA2040782 | single protein format | Scientific Literature | ||
| 15. | ALA2044628 | A | Inhibition of CYP3A5 at 10 uM | 1 | ALA2040782 | single protein format | Scientific Literature | ||
| 16. | ALA2390070 | A | Inhibition of CYP3A5 in human liver microsomes using midazolam as substrate by LC-MS/MS analysis | Homo sapiens | 4 | ALA2384956 | microsome format | Scientific Literature | |
| 17. | ALA3266607 | A | Inhibition of CYP3A5 (unknown origin) | Homo sapiens | 1 | ALA3259553 | single protein format | Scientific Literature | |
| 18. | ALA3266611 | A | Time-dependent inhibition of CYP3A5 (unknown origin) | Homo sapiens | 1 | ALA3259553 | single protein format | Scientific Literature | |
| 19. | ALA3388983 | A | Drug metabolism assessed as CYP3A5 (unknown origin)-mediated compound formation at 10 uM incubated for 60 mins in presence of NADPH by uHPLC-MS/MS method | Homo sapiens | 2 | ALA3351404 | single protein format | Scientific Literature | |
| 20. | ALA3387918 | A | Activity at human CYP3A5 assessed as enzyme-mediated drug metabolism | Homo sapiens | 1 | ALA3352375 | single protein format | Scientific Literature |
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