# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA650908 | B | Binding affinity towards CXCR3 receptor | 1 | single protein format | Scientific Literature | |||
2. | ALA828091 | B | Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK293 cells using [125I]CXCL10 as radioligand | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
3. | ALA836003 | F | Inhibition of CX3C chemokine receptor 3 mediated calcium release | Homo sapiens | 1 | assay format | Scientific Literature | ||
4. | ALA862999 | F | Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5 | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
5. | ALA863000 | F | Inhibition of CXCL10 (IP-10)-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5 | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
6. | ALA863001 | F | Inhibition of CXCL11-induced CXCR3 mediated T-cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
7. | ALA912822 | B | Inhibition of CXCR3 receptor at 2 to 20 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA905958 | F | Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assay | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
9. | ALA905961 | F | Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assay at 10 uM | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
10. | ALA888985 | B | Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMC | Homo sapiens | 47 | assay format | Scientific Literature | ||
11. | ALA888986 | F | Antagonist activity at human CXCR3 assessed as inhibition of MIG-induced calcium mobilization | Homo sapiens | 1 | assay format | Scientific Literature | ||
12. | ALA888990 | B | Displacement of [125I] ITAC from the CXCR3 receptor | Homo sapiens | 1 | single protein format | Scientific Literature | ||
13. | ALA888991 | F | Inhibition of IP10-induced CXCR3 mediated cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
14. | ALA888992 | F | Inhibition of ITAC-induced CXCR3 mediated cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
15. | ALA888993 | F | Inhibition of MIG-induced CXCR3 mediated cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
16. | ALA888994 | F | Antagonist activity at human CXCR3 assessed as inhibition of ITAC-induced calcium mobilization | Homo sapiens | 1 | assay format | Scientific Literature | ||
17. | ALA942022 | B | Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Homo sapiens | 27 | cell membrane format | Scientific Literature | ||
18. | ALA942023 | B | Inhibition of human CXCR3 expressed in CHO membrane at 10 uM by ITAC-stimulated GTP gammaS assay | Homo sapiens | 2 | cell membrane format | Scientific Literature | ||
19. | ALA928749 | F | Antagonist activity at human CXCR3 by [35S]GTP-gamma-S binding assay | Homo sapiens | 17 | assay format | Scientific Literature | ||
20. | ALA928937 | B | Displacement of [125I]IP-10 from CXCR3 receptor expressed in human PBMC in RPMI-1640 buffer supplemented with 0.5% BSA | 11 | assay format | Scientific Literature |