| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA650908 | B | Binding affinity towards CXCR3 receptor | 1 | single protein format | Scientific Literature | |||
| 2. | ALA828091 | B | Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK293 cells using [125I]CXCL10 as radioligand | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 3. | ALA836003 | F | Inhibition of CX3C chemokine receptor 3 mediated calcium release | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA862999 | F | Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5 | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 5. | ALA863000 | F | Inhibition of CXCL10 (IP-10)-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5 | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA863001 | F | Inhibition of CXCL11-induced CXCR3 mediated T-cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA912822 | B | Inhibition of CXCR3 receptor at 2 to 20 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA905958 | F | Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assay | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
| 9. | ALA905961 | F | Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTP-gamma-S binding assay at 10 uM | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 10. | ALA888985 | B | Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMC | Homo sapiens | 47 | assay format | Scientific Literature | ||
| 11. | ALA888986 | F | Antagonist activity at human CXCR3 assessed as inhibition of MIG-induced calcium mobilization | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA888990 | B | Displacement of [125I] ITAC from the CXCR3 receptor | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA888991 | F | Inhibition of IP10-induced CXCR3 mediated cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA888992 | F | Inhibition of ITAC-induced CXCR3 mediated cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA888993 | F | Inhibition of MIG-induced CXCR3 mediated cell migration | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA888994 | F | Antagonist activity at human CXCR3 assessed as inhibition of ITAC-induced calcium mobilization | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA2032961 | B | Inhibition of CXCR3 at 1 uM | 1 | single protein format | Scientific Literature | |||
| 18. | ALA1810318 | B | Ex vivo receptor occupancy of CXCR3 in human blood assessed as inhibition of ITAC binding after 1 hr by flow cytometry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 19. | ALA1810319 | B | Displacement of radiolabeled CXCL11 from human CXCR3 expressed in CHO cells by scintillation proximity assay | Homo sapiens | 52 | cell-based format | Scientific Literature | ||
| 20. | ALA1810320 | F | Antagonist activity at human CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assay | Homo sapiens | 52 | cell-based format | Scientific Literature |
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