# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA691020 | F | Activity was determined for the compound against the Mu opioid receptor by GTPgammaS functional assay using recombinant HEK293 cells. | 10 | ALA1147615 | cell-based format | Scientific Literature | ||
2. | ALA691172 | F | Activity was determined for the compound against the Mu opioid receptor by GTPgammaS functional assay using recombinant HEK293 cells; ND: Not determined | Homo sapiens | 5 | ALA1147615 | cell-based format | Scientific Literature | |
3. | ALA691173 | F | Activity was determined for the compound against the Mu opioid receptor by GTPgammaS functional assay using recombinant HEK293 cells; PA: Partial antagonist | Homo sapiens | 3 | ALA1147615 | cell-based format | Scientific Literature | |
4. | ALA878507 | F | Ratio of IC50 of morpholine (agonist) after 10 min of incubation along with compound (antagonist) and IC50 of agonist in absence of compound for mu opioid receptor at 1 uM in MVD assay | Mus musculus | 5 | ALA1123840 | assay format | Scientific Literature | |
5. | ALA746681 | B | Inhibition against mu receptor from displacement studies using 0.5 nM [3H]-DAMGO in rhesus monkey cortex membrane | Cercopithecidae | 22 | ALA1127360 | cell membrane format | Scientific Literature | |
6. | ALA747703 | F | Agonistic activity against human opioid Mu receptor transfected into Chinese hamster ovary (CHO) cells using [3H]-DAMGO as radioligand | 5 | ALA1131901 | cell-based format | Scientific Literature | ||
7. | ALA747704 | B | Binding affinity towards human opioid Mu receptor transfected into Chinese hamster ovary (CHO) cells using [3H]DAMGO as radioligand | 5 | ALA1131901 | cell-based format | Scientific Literature | ||
8. | ALA747705 | F | Agonistic activity against human opioid Delta receptor transfected into Chinese hamster ovary (CHO) cells using [3H]Cl-DPDPE as radioligand | 1 | ALA1131901 | cell-based format | Scientific Literature | ||
9. | ALA747706 | F | Agonistic activity against human opioid Mu receptor transfected into Chinese hamster ovary (CHO) cells using [3H]DAMGO as radioligand | 4 | ALA1131901 | cell-based format | Scientific Literature | ||
10. | ALA747707 | B | Displacement of [3H]naloxone from human mu opioid receptor | Homo sapiens | 14 | ALA1131838 | single protein format | Scientific Literature | |
11. | ALA747708 | B | Affinity for human mu opioid receptor was determined from competition binding curves using [3H]naloxone; ND means not determined | 1 | ALA1131838 | single protein format | Scientific Literature | ||
12. | ALA744603 | B | In vitro binding affinity towards mu opioid receptors was determined using [3H][p-Cl-Phe]- 4] DPDPE or [3H]deltorphin II | 9 | ALA1131989 | single protein format | Scientific Literature | ||
13. | ALA744604 | B | Compound was tested for binding affinity against mu opioid receptor binding assay | 2 | ALA1131909 | single protein format | Scientific Literature | ||
14. | ALA872654 | B | Tested in vitro for binding affinity against mu opioid receptor | 4 | ALA1126961 | single protein format | Scientific Literature | ||
15. | ALA749648 | F | Agonistic activity against Opioid receptor mu 1 in Chinese hamster ovary membranes | Cricetulus griseus | 4 | ALA1149134 | cell membrane format | Scientific Literature | |
16. | ALA749649 | F | Binding ability against Opioid receptor mu 1 by stimulating the [35S]GTP-gamma-S radioligand in Chinese hamster ovary membranes | Cricetulus griseus | 4 | ALA1149134 | cell membrane format | Scientific Literature | |
17. | ALA749650 | B | Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of Chinese hamster ovary membrane | Cricetulus griseus | 13 | ALA1149134 | assay format | Scientific Literature | |
18. | ALA749651 | F | Maximal activation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranes | 2 | ALA1135663 | assay format | Scientific Literature | ||
19. | ALA749652 | F | Percent stimulation of [35S]GTP-gamma-S, binding in recombinant human Opioid receptor mu 1 transfected into CHO cells | 2 | ALA1144921 | cell-based format | Scientific Literature | ||
20. | ALA749653 | F | Percent stimulation of [35S]GTP-gamma-S, binding in recombinant human Opioid receptor mu 1 transfected into CHO cells: Antagonist activity | 2 | ALA1144921 | cell-based format | Scientific Literature |