| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA757347 | F | Effective agonist concentration to the human Orexin receptor type 2 was determined using the Xlfit program | 79 | ALA1148480 | assay format | Scientific Literature | ||
| 2. | ALA757348 | B | Inhibitory concentration against human orexin-2 receptor (hOX2R) | 29 | ALA1136503 | single protein format | Scientific Literature | ||
| 3. | ALA757349 | B | Compound was evaluated for its binding affinity towards Orexin receptor type 2 | 1 | ALA1134731 | single protein format | Scientific Literature | ||
| 4. | ALA840218 | B | Binding affinity towards human orexin receptor type 2 was determined using [125I]-Orexin A as radio ligand | Homo sapiens | 30 | ALA1137156 | single protein format | Scientific Literature | |
| 5. | ALA835462 | F | Antagonistic activity towards intracellular calcium levels in cells expressing Orexin receptor type 2 | Homo sapiens | 5 | ALA1137156 | cell-based format | Scientific Literature | |
| 6. | ALA857325 | F | Agonist activity against human orexin 2 receptor; EC50; nM | Homo sapiens | 61 | ALA1145783 | assay format | Scientific Literature | |
| 7. | ALA932891 | B | Displacement of [3H](S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2R expressed in CHO cells | Homo sapiens | 20 | ALA1143219 | cell-based format | Scientific Literature | |
| 8. | ALA932892 | F | Antagonist activity at human OX2R expressed in CHOK1 cells assessed as effect on calcium mobilization | Homo sapiens | 19 | ALA1143219 | cell-based format | Scientific Literature | |
| 9. | ALA1007893 | F | Antagonist activity at human OX2 receptor expressed in CHO cells assessed as inhibition of receptor-mediated calcium response by FLIPR | Homo sapiens | 1 | ALA1140924 | cell-based format | Scientific Literature | |
| 10. | ALA1007898 | F | Antagonist activity at human OX2 receptor | Homo sapiens | 29 | ALA1140924 | assay format | Scientific Literature | |
| 11. | ALA1007903 | B | Binding affinity to OX2 receptor | 18 | ALA1140924 | single protein format | Scientific Literature | ||
| 12. | ALA1007909 | B | Inhibition of OX2 receptor | 37 | ALA1140924 | single protein format | Scientific Literature | ||
| 13. | ALA1007911 | F | Antagonist activity at OX2 receptor by FLIPR | 13 | ALA1140924 | assay format | Scientific Literature | ||
| 14. | ALA998534 | F | Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assay | Homo sapiens | 15 | ALA1152230 | cell-based format | Scientific Literature | |
| 15. | ALA998535 | F | Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of ATP-stimulated calcium release by FLIPR assay | Homo sapiens | 15 | ALA1152230 | cell-based format | Scientific Literature | |
| 16. | ALA998536 | F | Agonist activity at human OX2 receptor expressed in HEK293 cells assessed as effect on human orexin-A-stimulated calcium release by FLIPR assay | Homo sapiens | 15 | ALA1152230 | cell-based format | Scientific Literature | |
| 17. | ALA1006173 | F | Inhibition of human OX2 receptor expressed in CHO cells assessed as intercellular calcium mobilization by FLIPR assay | Homo sapiens | 37 | ALA1143438 | cell-based format | Scientific Literature | |
| 18. | ALA973408 | B | Binding affinity to OX2 receptor | 6 | ALA1136898 | single protein format | Scientific Literature | ||
| 19. | ALA1099401 | F | Antagonist activity at human OX2 receptor expressed in CHO cells assessed as inhibition of calcium mobilization by FLIPR assay | Homo sapiens | 15 | ALA1154972 | cell-based format | Scientific Literature | |
| 20. | ALA1109766 | B | Binding affinity to OX2 receptor by radioligand displacement assay | 7 | ALA1156317 | single protein format | Scientific Literature |
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