| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA815442 | B | Inhibition of human V1A vasopressin receptor | Homo sapiens | 5 | ALA1134625 | single protein format | Scientific Literature | |
| 2. | ALA815444 | B | In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membrane | 4 | ALA1131757 | assay format | Scientific Literature | ||
| 3. | ALA815445 | B | In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membrane at 10 uM | 1 | ALA1131757 | assay format | Scientific Literature | ||
| 4. | ALA819416 | B | Ability to displace [3H]arginine vasopressin in cloned human V1a receptor | Homo sapiens | 10 | ALA1136360 | single protein format | Scientific Literature | |
| 5. | ALA819417 | B | Binding affinity measured by inhibition of 3[H] AVP binding to cloned human vasopressin V1a receptor | 16 | ALA1146639 | single protein format | Scientific Literature | ||
| 6. | ALA819418 | B | Binding affinity measured by inhibition of 3[H] AVP binding to cloned human vasopressin V1a receptor (Compound 7o) | 1 | ALA1146639 | single protein format | Scientific Literature | ||
| 7. | ALA819419 | B | Binding affinity towards VIa receptor | 1 | ALA1136603 | single protein format | Scientific Literature | ||
| 8. | ALA819420 | B | Binding affinity towards human V1a receptors | 1 | ALA1136603 | single protein format | Scientific Literature | ||
| 9. | ALA881932 | F | Inhibition of vasopressin induced calcium immobilization in human V1a receptor expressing cells | Homo sapiens | 6 | ALA1136360 | assay format | Scientific Literature | |
| 10. | ALA884682 | F | Inhibition of vasopressin induced calcium immobilization in human V1a receptor expressing cells; ND= Not determined | Homo sapiens | 5 | ALA1136360 | assay format | Scientific Literature | |
| 11. | ALA819421 | B | In vitro binding affinity to human V1a receptor | Homo sapiens | 9 | ALA1133322 | single protein format | Scientific Literature | |
| 12. | ALA819422 | B | In vitro binding affinity to human V1a receptor; not tested | Homo sapiens | 7 | ALA1133322 | single protein format | Scientific Literature | |
| 13. | ALA819423 | B | In vitro binding affinity to human V1a receptor; Not tested | 1 | ALA1133322 | single protein format | Scientific Literature | ||
| 14. | ALA819424 | F | Evaluated for intracellular calcium mobilization in HEK- 293 cells transfected to express human vasopressin V1a receptor (Compound 7o) | 1 | ALA1146639 | cell-based format | Scientific Literature | ||
| 15. | ALA820271 | F | Evaluated for intracellular calcium mobilization in HEK293 cells transfected to express human vasopressin V1a receptor | 16 | ALA1146639 | cell-based format | Scientific Literature | ||
| 16. | ALA820272 | B | Inhibition of [3H]Arg-vasopressin binding to recombinant human vasopressin V1a receptor | Homo sapiens | 11 | ALA1134932 | single protein format | Scientific Literature | |
| 17. | ALA820273 | B | In vitro inhibitory concentration against [3H]AVP binding to cloned human vasopressin V1a receptor | 17 | ALA1146774 | single protein format | Scientific Literature | ||
| 18. | ALA820274 | B | Ability to displace [3H]arginine vasopressin in cloned human V1a receptor | Homo sapiens | 1 | ALA1136360 | single protein format | Scientific Literature | |
| 19. | ALA881115 | B | Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptor at 1000 nM | Homo sapiens | 1 | ALA1146755 | single protein format | Scientific Literature | |
| 20. | ALA820275 | B | Inhibition of [3H]Arg-vasopressin binding to recombinant human vasopressin V1a receptor at 0.1 uM | Homo sapiens | 3 | ALA1134932 | single protein format | Scientific Literature |
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