# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA895396 | B | Displacement of [125I]-[Nle,8,18 Tyr34]-hPTH(1-34) from human recombinant PTH1R expressed in HEK293 cells | Homo sapiens | 26 | ALA1148813 | cell-based format | Scientific Literature | |
2. | ALA895397 | F | Antagonist activity at human wild type PTH1 receptor expressed in SaOS2 cells assessed as inhibition of PTHrP (1-34)-stimulated cAMP production at 3 uM | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
3. | ALA895399 | F | Antagonist activity at human recombinant PTH2 receptor expressed in CHOK1 cells assessed as inhibition of TIP (1-39)-stimulated cAMP production at 10 uM | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
4. | ALA895400 | B | Displacement of [125I]-[Nle,8,18 Tyr34]-hPTH(1-34) from human recombinant PTH1R expressed in HEK293 cells at 1 uM | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
5. | ALA895401 | B | Displacement of [125I]-[Nle,8,18 Tyr34]-hPTH(1-34) from human recombinant PTH1R expressed in HEK293 cells at 30 uM | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
6. | ALA895402 | B | Displacement of [125I]-[Nle,8,18 Tyr34]-hPTH(1-34) from human recombinant PTH1R expressed in HEK293 cells at 10 uM | Homo sapiens | 2 | ALA1148813 | cell-based format | Scientific Literature | |
7. | ALA895403 | F | Activity at human PTH1 receptor expressed in SaOS2 cells assessed as cAMP production upto 10 uM | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
8. | ALA895404 | F | Antagonist activity at human recombinant PTH1 receptor expressed in HEK293 cells assessed as inhibition of PTH(1-34)-stimulated cAMP production | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
9. | ALA895406 | F | Antagonist activity at human wild type PTH1 receptor expressed in SaOS2 cells assessed as inhibition of PTHrP (1-34)-stimulated cAMP production | Homo sapiens | 1 | ALA1148813 | cell-based format | Scientific Literature | |
10. | ALA944461 | F | Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of intracellular calcium mobilization | Homo sapiens | 1 | ALA1156459 | cell-based format | Scientific Literature | |
11. | ALA944462 | F | Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter assay | Homo sapiens | 8 | ALA1156459 | cell-based format | Scientific Literature | |
12. | ALA944464 | F | Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formation | Homo sapiens | 8 | ALA1156459 | cell-based format | Scientific Literature | |
13. | ALA944465 | B | Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor expressed in HKRK-B28 cells | 9 | ALA1156459 | cell-based format | Scientific Literature | ||
14. | ALA944466 | B | Binding affinity to PTH/PTH-related peptide receptor expressed in HKRK-B28 cells | 1 | ALA1156459 | cell-based format | Scientific Literature | ||
15. | ALA945433 | F | Antagonist activity at human PTH/PTH-related peptide receptor expressed in human CL0153 cells assessed as inhibition of DPC-AJ1951-induced cAMP production | Homo sapiens | 1 | ALA1156459 | cell-based format | Scientific Literature | |
16. | ALA945434 | F | Antagonist activity at human PTH/PTH-related peptide receptor expressed in human SaOS2 assessed as inhibition of DPC-AJ1951-induced cAMP production | Homo sapiens | 1 | ALA1156459 | cell-based format | Scientific Literature | |
17. | ALA945435 | F | Antagonist activity at PTH/PTH-related peptide receptor expressed in HKRK-B28 cells assessed as inhibition of DPC-AJ1951-induced cAMP production | 1 | ALA1156459 | cell-based format | Scientific Literature | ||
18. | ALA945436 | F | Antagonist activity at PTH/PTH-related peptide receptor expressed in HKRK-B28 cells assessed as inhibition of parathyroid hormone (1 to 34)-induced cAMP production | 1 | ALA1156459 | cell-based format | Scientific Literature | ||
19. | ALA945456 | B | Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor expressed in HKRK-B28 cells in presence of SW106 | 1 | ALA1156459 | cell-based format | Scientific Literature | ||
20. | ALA1050759 | F | Agonist activity at PTHR | 1 | ALA1156009 | assay format | Scientific Literature |