# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA868780 | B | Binding affinity to VMAT2 | Homo sapiens | 1 | ALA1148600 | single protein format | Scientific Literature | |
2. | ALA931822 | B | Inhibition of monoamine transporter | 1 | ALA1143219 | single protein format | Scientific Literature | ||
3. | ALA953427 | B | Inhibition of monoamine transporter at 10 uM | 1 | ALA1150320 | single protein format | Scientific Literature | ||
4. | ALA1044344 | B | Binding affinity to VMAT2 | 1 | ALA1155310 | single protein format | Scientific Literature | ||
5. | ALA1068127 | B | Binding affinity to VMAT2 receptor | 5 | ALA1159052 | single protein format | Scientific Literature | ||
6. | ALA2089938 | B | Activity at vesicular monoamine transporter 2 at 10 uM | 1 | ALA2086249 | single protein format | Scientific Literature | ||
7. | ALA4202136 | B | Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 19 | ALA4196220 | cell-based format | Scientific Literature | |
8. | ALA4202137 | B | Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting method | Homo sapiens | 19 | ALA4196220 | cell-based format | Scientific Literature | |
9. | ALA4202138 | B | Binding affinity to human VMAT2 expressed in HEK293 cell membranes in presence of 2 mM Mg-ATP by scintillation counting method | Homo sapiens | 3 | ALA4196220 | cell-based format | Scientific Literature | |
10. | ALA4202139 | B | Binding affinity to human VMAT2 expressed in HEK293 cell membranes assessed as observed associate rate combatant at 14 to 22 nM in presence of 2 mM Mg-ATP by scintillation counting method | Homo sapiens | 1 | ALA4196220 | cell-based format | Scientific Literature | |
11. | ALA4202140 | B | Binding affinity to human VMAT2 expressed in HEK293 cell membranes assessed as observed associate rate constant at 24 to 28 nM in presence of 2 mM Mg-ATP by scintillation counting method | Homo sapiens | 1 | ALA4196220 | cell-based format | Scientific Literature | |
12. | ALA4202141 | B | Binding affinity to human VMAT2 expressed in HEK293 cell membranes assessed as half life at 24 to 28 nM in presence of 2 mM Mg-ATP by scintillation counting method | Homo sapiens | 1 | ALA4196220 | cell-based format | Scientific Literature | |
13. | ALA4202142 | B | Binding affinity to human VMAT2 expressed in HEK293 cell membranes assessed as half life at 14 to 22 nM in presence of 2 mM Mg-ATP by scintillation counting method | Homo sapiens | 1 | ALA4196220 | cell-based format | Scientific Literature | |
14. | ALA4202143 | B | Binding affinity to human VMAT2 expressed in HEK293 cell membranes by scintillation counting method based saturation binding assay | Homo sapiens | 3 | ALA4196220 | cell-based format | Scientific Literature | |
15. | ALA4202144 | B | Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 19 | ALA4196220 | cell-based format | Scientific Literature | |
16. | ALA4202145 | B | Inhibition of human VMAT2 expressed in HEK293 cell membranes assessed as reduction in [3H[-5HT uptake pre-incubated for 10 mins before [3H[-5HT addition and measured after 6 mins | Homo sapiens | 19 | ALA4196220 | cell-based format | Scientific Literature | |
17. | ALA4621413 | B | Inhibition of VMAT2 (unknown origin) | Homo sapiens | 1 | ALA4619774 | single protein format | Scientific Literature | |
18. | ALA4668878 | A | Inhibition of VMAT2 (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | ALA4665701 | single protein format | Scientific Literature | |
19. | ALA4883047 | B | Transporter, Monoamine Eurofins-Panlabs radioligand binding assay | Oryctolagus cuniculus | 2 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
20. | ALA5163326 | B | Inhibition of vesicular monoamine transporter 2 (unknown origin) | Homo sapiens | 1 | ALA5154826 | single protein format | Scientific Literature |