# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA644077 | B | Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranes | 6 | ALA1126929 | cell membrane format | Scientific Literature | ||
2. | ALA652389 | F | Antagonistic activity against beta-2 adrenergic receptor as inhibition of vasopressor response in rats | Rattus norvegicus | 7 | ALA1122842 | assay format | Scientific Literature | |
3. | ALA652393 | B | Displacement of [3H]DHA (Dihydroalprenolol) from beta-2 adrenergic receptor in rat brain | Rattus norvegicus | 2 | ALA1124042 | tissue-based format | Scientific Literature | |
4. | ALA652395 | B | Binding affinity against beta-2 adrenergic receptor in rat brain using [3H]DHA | Rattus norvegicus | 2 | ALA1123363 | tissue-based format | Scientific Literature | |
5. | ALA652396 | B | Binding affinity against the beta-2 adrenergic receptor using [3H]- DHA | Rattus norvegicus | 1 | ALA1123363 | single protein format | Scientific Literature | |
6. | ALA652286 | B | Compound was evaluated for its binding affinity towards Beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 uM) | 3 | ALA1125527 | cell membrane format | Scientific Literature | ||
7. | ALA652288 | B | Binding affinity against beta-2 adrenergic receptor in rat brain using [3H]DHA | Rattus norvegicus | 1 | ALA1123363 | tissue-based format | Scientific Literature | |
8. | ALA652289 | F | Inhibition of spontaneous contractions in isolated rat uterus | Rattus norvegicus | 7 | ALA1145008 | tissue-based format | Scientific Literature | |
9. | ALA652292 | B | Apparent dissociation constant towards beta-2 adrenergic receptor in rat lung membranes using (2-6)x10E-9M of [3AH]-DHA in the presence or absence of 10e-5 M (+/-) propranolol. | Rattus norvegicus | 10 | ALA1123880 | cell membrane format | Scientific Literature | |
10. | ALA820267 | B | Displacement of [125 I ] iodocyanopindolol from cloned beta-2 receptor expressed in CHO cells | Rattus norvegicus | 1 | ALA1126642 | cell-based format | Scientific Literature | |
11. | ALA819428 | F | Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contraction | Rattus norvegicus | 19 | ALA1134410 | assay format | Scientific Literature | |
12. | ALA895334 | F | Vasodilating activity against phenylephrine-induced contraction in rat thoracic aorta in presence of 1H-[1,2,4]oxadiazolo-[4,3-a]quinoxalin-1-one | Rattus norvegicus | 3 | ALA1148806 | tissue-based format | Scientific Literature | |
13. | ALA895341 | F | Vasodilating activity against phenylephrine-induced contractions in rat thoracic aorta at 100 uM in presence of 1H-[1,2,4]oxadiazolo-[4,3-a]quinoxalin-1-one | Rattus norvegicus | 2 | ALA1148806 | tissue-based format | Scientific Literature | |
14. | ALA895342 | F | Vasodilating activity against phenylephrine-induced contractions in rat thoracic aorta | Rattus norvegicus | 6 | ALA1148806 | tissue-based format | Scientific Literature | |
15. | ALA895344 | F | Vasodilating activity in rat thoracic aorta on phenylephrine-induced contraction at 100 uM | Rattus norvegicus | 1 | ALA1148806 | tissue-based format | Scientific Literature | |
16. | ALA1259775 | B | Binding affinity to rat adrenergic beta2 receptor | Rattus norvegicus | 3 | ALA1255169 | single protein format | Scientific Literature | |
17. | ALA1804513 | F | Agonist activity beta2-adrenergic receptor in rat ventricular myocytes assessed as cell contraction following electrical stimulation by optical edge tracking method using photodiode array | Rattus norvegicus | 9 | ALA1800026 | cell-based format | Scientific Literature | |
18. | ALA1804514 | F | Agonist activity beta2-adrenergic receptor in rat ventricular myocytes assessed as cell contraction following electrical stimulation by optical edge tracking method using photodiode array in presence of receptor antagonist ICI 118551 | Rattus norvegicus | 1 | ALA1800026 | cell-based format | Scientific Literature | |
19. | ALA1804515 | F | Agonist activity beta2-adrenergic receptor in rat ventricular myocytes assessed as cell contraction following electrical stimulation by optical edge tracking method using photodiode array in presence of receptor agonist zinterol | Rattus norvegicus | 1 | ALA1800026 | cell-based format | Scientific Literature | |
20. | ALA2415468 | B | Antagonist activity at alpha2 adrenoreceptor in rat brain cortical membranes assessed as inhibition of [3H]-RX821002 binding to receptor after 45 mins by competition assay in absence of GTP | Rattus norvegicus | 2 | ALA2412990 | cell membrane format | Scientific Literature |