# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA645314 | F | Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membrane | Sus scrofa | 9 | ALA1123293 | cell membrane format | Scientific Literature | |
2. | ALA817084 | F | Agonistic activity of the V2 system was evaluated bythe adenylate cyclase activity in LLCPK cells at a concentration of 10E-7 M; No activity | 1 | ALA1126290 | cell-based format | Scientific Literature | ||
3. | ALA817085 | F | Antagonistic activity of the V2 system was evaluated bythe adenylate cyclase activity in LLCPK cells at a concentration of 10E-7 M; No activity | 1 | ALA1126290 | cell-based format | Scientific Literature | ||
4. | ALA817086 | B | Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cells | 2 | ALA1129881 | cell-based format | Scientific Literature | ||
5. | ALA817087 | B | Inhibition constant for [3H]LVP binding to medullary membranes of pig kidney | 9 | ALA1124391 | tissue-based format | Scientific Literature | ||
6. | ALA817088 | F | Binding affinity towards V2-receptor in LLCPK cells | 1 | ALA1126290 | cell-based format | Scientific Literature | ||
7. | ALA817089 | B | Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney | 9 | ALA1124391 | assay format | Scientific Literature | ||
8. | ALA815389 | B | Compound was tested for binding affinity against V2 vasopressin receptor in pig renal medullary membrane preparations using tritiated LVP. | 7 | ALA1123377 | cell membrane format | Scientific Literature | ||
9. | ALA815390 | B | Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations. | 4 | ALA1123377 | cell membrane format | Scientific Literature | ||
10. | ALA815391 | F | Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations; e=Partial agonist with a relative Vmax of 14%. | 1 | ALA1123377 | cell membrane format | Scientific Literature | ||
11. | ALA815392 | B | Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations; nd=Not determined | 2 | ALA1123377 | cell membrane format | Scientific Literature | ||
12. | ALA818338 | F | Agonistic activity of the V2 system (Vasopressin V2 receptor) was evaluated bythe adenylate cyclase activity in LLCPK cells at a concentration of 10E-7 M; No activity | 1 | ALA1126290 | cell-based format | Scientific Literature | ||
13. | ALA818339 | F | Antagonistic activity of the V2 system (Vasopressin V2 receptor) was evaluated bythe adenylate cyclase activity in LLCPK cells at a concentration of 10E-7 M; No activity | 1 | ALA1126290 | cell-based format | Scientific Literature | ||
14. | ALA818340 | B | In vitro antagonist activity was measured by inhibition of binding of [3H]LVP to renal medullary membrane preparation in pig | 1 | ALA1124168 | tissue-based format | Scientific Literature | ||
15. | ALA818341 | B | Inhibition constant for [3H]LVP binding to medullary membranes of pig kidney of Vasopressin V2 receptor | Sus scrofa | 11 | ALA1124391 | assay format | Scientific Literature | |
16. | ALA818342 | B | Vasopressin V2 receptor binding affinity measured by competition with tritiated LVP lysine vasopressin in pig renal medullary preparation | 4 | ALA1124075 | single protein format | Scientific Literature | ||
17. | ALA820052 | B | Binding affinity towards Vasopressin V2 receptor in LLCPK cells | 1 | ALA1126290 | cell-based format | Scientific Literature | ||
18. | ALA820053 | B | Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor) | 9 | ALA1124391 | assay format | Scientific Literature | ||
19. | ALA820054 | B | Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor); NT=Not tested | 2 | ALA1124391 | assay format | Scientific Literature | ||
20. | ALA820055 | B | Inhibition of LVP-sensitive adenylate cyclase in a pig renal medullary preparation | 4 | ALA1124075 | tissue-based format | Scientific Literature |