| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA809058 | B | Binding affinity against Sodium/glucose co-transporter of isolated renal brush border membranes. | Homo sapiens | 19 | ALA1132925 | assay format | Scientific Literature | |
| 2. | ALA834934 | F | In vitro inhibition of Na-dependent [14C]AMG uptake in CHO-K1 cells expressing human sodium glucose co-transporter 1 | Homo sapiens | 23 | ALA1137899 | cell-based format | Scientific Literature | |
| 3. | ALA863284 | B | Inhibitory activity towards human SGLT1 expressed in CHO-K1 cells | Homo sapiens | 6 | ALA1141232 | cell-based format | Scientific Literature | |
| 4. | ALA863287 | B | Inhibitory activity towards human SGLT1 expressed in CHO-K1 cells at 10 uM | Homo sapiens | 7 | ALA1141232 | cell-based format | Scientific Literature | |
| 5. | ALA869549 | B | Inhibitory activity against SGLT1 expressed in CHO-K1 cells | Homo sapiens | 15 | ALA1139015 | cell-based format | Scientific Literature | |
| 6. | ALA868396 | B | Inhibition of SGLT1 expressed in CHO-K1 cells at 10 uM | Homo sapiens | 9 | ALA1139015 | cell-based format | Scientific Literature | |
| 7. | ALA892510 | B | Inhibition of human SGLT1 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake at 50 uM | Homo sapiens | 9 | ALA1147913 | cell-based format | Scientific Literature | |
| 8. | ALA892512 | B | Inhibition of human SGLT1 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake | Homo sapiens | 3 | ALA1147913 | cell-based format | Scientific Literature | |
| 9. | ALA947998 | B | Inhibition of human SGLT1 expressed in CHO cells assessed as inhibition of [14C]AMG accumulation | Homo sapiens | 5 | ALA1142359 | cell-based format | Scientific Literature | |
| 10. | ALA978802 | B | Reversal of inhibition of human SGLT1 expressed in xenopus laevis oocyte by measuring inhibition of methyl-alpha-D-[14C]glucopyranoside uptake after 1 hr assessed concentration required for 50% protective high affinity in presence of methyl-alpha-D-glucopyranoside relative to control | Homo sapiens | 2 | ALA1156499 | assay format | Scientific Literature | |
| 11. | ALA978803 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 1 hr relative to control | Homo sapiens | 11 | ALA1156499 | assay format | Scientific Literature | |
| 12. | ALA978804 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as decrease in amount of SGLT1 protein level in oocyte plasma membrane at 75 pmol after 1 hr by Western blotting relative to control | Homo sapiens | 1 | ALA1156499 | cell membrane format | Scientific Literature | |
| 13. | ALA978805 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as decrease in phlorizin-induced capacitance at 75 pmol after 1 hr by relative to control | Homo sapiens | 1 | ALA1156499 | assay format | Scientific Literature | |
| 14. | ALA978806 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 1 hr in presence of botulinum toxin B relative to control | Homo sapiens | 1 | ALA1156499 | assay format | Scientific Literature | |
| 15. | ALA974292 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 1 hr in presence of brefeldin A relative to control | Homo sapiens | 1 | ALA1156499 | assay format | Scientific Literature | |
| 16. | ALA974293 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 9 hrs relative to control | Homo sapiens | 1 | ALA1156499 | assay format | Scientific Literature | |
| 17. | ALA974294 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake after 1 hrs | Homo sapiens | 4 | ALA1156499 | assay format | Scientific Literature | |
| 18. | ALA974295 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 1 hr in presence of mannitol relative to control | Homo sapiens | 1 | ALA1156499 | assay format | Scientific Literature | |
| 19. | ALA974296 | B | Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 1 hr in presence of sorbitol relative to control | Homo sapiens | 1 | ALA1156499 | assay format | Scientific Literature | |
| 20. | ALA974297 | B | Reversal of inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake at 75 pmol after 1 hr in presence of D-glucose relative to control | Homo sapiens | 2 | ALA1156499 | assay format | Scientific Literature |
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