| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3615705 | B | Inhibition of Nav2.1 channel (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA4321987 | B | Inhibition of human Nav1.7 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 3. | ALA4322019 | B | Binding affinity to human recombinant Nav1.7 by radioligand binding assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 4. | ALA4481270 | B | Inhibition of human NaV1.7 expressed in HEK293 cells at 1 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA4630241 | B | Inhibition of human NaV1.7 at 100 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 6. | ALA4720268 | B | Inhibition of human Nav1.7 expressed in HEK293 cells up to 1 uM incubated for 30 mins by FLIPRTetra fluorescent membrane potential assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA5055691 | B | Displacement of [3H]GX-545 Nav1.7 (unknown origin) expressed in HEK cells by liquid scintillation counting based radioligand competition assay | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 8. | ALA5055692 | B | Inhibition of human Nav1.7 expressed in HEK293 cells incubated for 1 hr in presence of veratridine by sodium influx assay | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 9. | ALA5055697 | B | Inhibition of full length human Nav1.7 expressed in HEK cells by whole cell voltage clamp analysis | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 10. | ALA5055729 | B | Inhibition of human Nav1.7 expressed in HEK293 cells assessed as fold change incubated for 1 hr in presence of BSA by sodium influx assay | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 11. | ALA5123729 | B | Inhibition of Nav1.7 (unknown origin) in resting condition at 30 uM by whole cell patch clamp electrophysiology relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA5123732 | B | Inhibition of Nav1.7 (unknown origin) in half-inactivated condition at 30 uM by whole cell patch clamp electrophysiology relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA5123772 | B | Inhibition of Nav1.7 (unknown origin) in resting condition at 1 uM by whole cell patch clamp electrophysiology relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA5123773 | B | Inhibition of Nav1.7 (unknown origin) in half-inactivated condition at 1 uM by whole cell patch clamp electrophysiology relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA5131327 | B | Inhibition of human Nav1.7 expressed in HEK293 cells at -120 mV holding potential by automated patch clamp electrophysiology recording | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA5147694 | B | Inhibition of recombinant human Nav 1.7 expressed in HEK293F cells incubated for 3 mins by FRET based membrane potential assay | Homo sapiens | 49 | cell membrane format | Scientific Literature | ||
| 17. | ALA5147703 | B | Inhibition of recombinant human Nav 1.7 expressed in HEK293F cells at -65 mV holding potential by Qpatch clamp electrophysiology method | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 18. | ALA5147781 | B | Inhibition of recombinant human Nav 1.7 expressed in HEK293F cells at -65 to 80 mV holding potential by manual voltage clamp electrophysiology method | Homo sapiens | 1 | cell-based format | Scientific Literature |
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