# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1048220 | Binding | Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assay | Homo sapiens | 22 | ALA1155971 | cell-based format | Scientific Literature | |
2. | ALA1048221 | Binding | Inhibition of human Nav1.7 channel expressed in HEK cells at 1 uM by FRET assay | Homo sapiens | 32 | ALA1155971 | cell-based format | Scientific Literature | |
3. | ALA1042688 | Binding | Inhibition of human Nav1.7 channel expressed in HEK293 cells by FRET assay | Homo sapiens | 26 | ALA1155991 | cell-based format | Scientific Literature | |
4. | ALA1042689 | Binding | Inhibition of human Nav1.7 channel expressed in HEK293 cells at 1 uM by FRET assay | Homo sapiens | 9 | ALA1155991 | cell-based format | Scientific Literature | |
5. | ALA971436 | Binding | Inhibition of human Nav1.7 expressed in HEK293 cells assessed as change in membrane potential using MP-red voltage sensitive dye at 10 uM | Homo sapiens | 5 | ALA1138611 | cell-based format | Scientific Literature | |
6. | ALA829428 | Binding | In vitro inhibitory concentration against Na v1.7 channel electrophysiology in inactivated state expressed in HEK293 cells using Voltage/Ion Probe Reader (VIPR) assay | Homo sapiens | 2 | ALA1140272 | cell-based format | Scientific Literature | |
7. | ALA826159 | Binding | In vitro inhibitory concentration against Na v1.7 channel electrophysiology in resting state expressed in HEK293 cells using Voltage/Ion Probe Reader (VIPR) assay | Homo sapiens | 1 | ALA1140272 | cell-based format | Scientific Literature | |
8. | ALA829086 | Binding | In vivo inhibitory concentration against Na v1.7 channel expressed in HEK293 cells using Voltage/Ion Probe Reader (VIPR) assay | Homo sapiens | 1 | ALA1140272 | organism-based format | Scientific Literature | |
9. | ALA829535 | Binding | In vitro inhibitory concentration against Na v1.7 channel expressed in HEK293 cells using Voltage/Ion Probe Reader (VIPR) assay | Homo sapiens | 25 | ALA1140272 | cell-based format | Scientific Literature | |
10. | ALA834889 | Functional | In vitro inhibitory concentration against Na v1.7 channel electrophysiology in resting state expressed in HEK293 cells using Voltage/Ion Probe Reader (VIPR) assay | Homo sapiens | 1 | ALA1140272 | cell-based format | Scientific Literature | |
11. | ALA834126 | Functional | Inhibitory constant against voltage-gated sodium channel Nav1.7 in electrophysiology assays (EP) | 26 | ALA1143509 | assay format | Scientific Literature | ||
12. | ALA874197 | Functional | In vitro inhibitory concentration against voltage-gated sodium channel Nav1.7 in voltage-ion-probe-reader (VIPR) assay | 48 | ALA1143509 | assay format | Scientific Literature | ||
13. | ALA866524 | Binding | Inhibition of peripheral nerve sodium channel NaV1.7 | Homo sapiens | 23 | ALA1138981 | single protein format | Scientific Literature | |
14. | ALA924068 | Binding | Blockade of human Nav1.7 by FRET assay | Homo sapiens | 43 | ALA1140675 | single protein format | Scientific Literature | |
15. | ALA923058 | Binding | Binding affinity at human inactive state Nav1.7 by whole cell electrophysiology | Homo sapiens | 1 | ALA1140675 | single protein format | Scientific Literature | |
16. | ALA923059 | Binding | Binding affinity at human resting state Nav1.7 by whole cell electrophysiology | Homo sapiens | 1 | ALA1140675 | single protein format | Scientific Literature | |
17. | ALA924359 | Binding | Inhibition of human sodium channel Nav1.7 by FRET assay | Homo sapiens | 24 | ALA1140523 | single protein format | Scientific Literature | |
18. | ALA944713 | Binding | Inhibition of human Nav1.7 channel at 3 uM | Homo sapiens | 4 | ALA1140726 | single protein format | Scientific Literature | |
19. | ALA944714 | Binding | Inhibition of human Nav1.7 channel at 1 uM | Homo sapiens | 4 | ALA1140726 | single protein format | Scientific Literature | |
20. | ALA944715 | Binding | Inhibition of human Nav1.7 channel at 10 uM | Homo sapiens | 2 | ALA1140726 | single protein format | Scientific Literature |