# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA818201 | F | Blockade of synaptosomal sodium channels, inhibition of [14C]guanidinium ion flux into CHO cells expressing Type II sodium channel | 3 | cell-based format | Scientific Literature | |||
2. | ALA818202 | F | Blockade of synaptosomal sodium channels, inhibition of [14C]guanidinium ion flux into CHO cells expressing Type II sodium channel | 1 | cell-based format | Scientific Literature | |||
3. | ALA843814 | B | Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channel | 41 | cell-based format | Scientific Literature | |||
4. | ALA1809308 | B | Inhibition of human voltage-gated sodium channel 1.2 expressed in human HEK293 cells at 10 uM by two-microelectrode voltage-clamp electrophysiology | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
5. | ALA1809309 | B | Inhibition of human voltage-gated sodium channel 1.2 expressed in HEK293 cells at 1 uM by two-microelectrode voltage-clamp electrophysiology | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
6. | ALA1809310 | B | Inhibition of human voltage-gated sodium channel 1.2 expressed in HEK293 cells at 100 nM by two-microelectrode voltage-clamp electrophysiology | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
7. | ALA931276 | B | Inhibition of human Nav1.2 channel expressed in HEK293 cells at -120 mV by patch clamp method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
8. | ALA931277 | B | Inhibition of human Nav1.2 channel expressed in HEK293 cells at -60 mV by patch clamp method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
9. | ALA926141 | B | Inhibition of inactivated human Nav1.2 sodium channel | Homo sapiens | 1 | single protein format | Scientific Literature | ||
10. | ALA2072611 | B | Inhibition of human NaV1.2 expressed in HEK293 cells at 10 uM using sodium currents elicited through depolarizing step from holding potential of -100 mV to +10 mV for 25 ms at 15 s intervals by whole cell patch clamp method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
11. | ALA1959244 | B | Inhibition of human voltage-gated sodium channel 1.2-mediated current expressed in HEK293 cells at -60 to +10 mV holding poteinitial at 1 uM after 5 mins by patch clamp electrophysiology | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
12. | ALA1959245 | B | Inhibition of human voltage-gated sodium channel 1.2-mediated current expressed in HEK293 cells at -60 to +10 mV holding poteinitial at 10 uM after 5 mins by patch clamp electrophysiology | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
13. | ALA1959246 | B | Reversible inhibition of human voltage-gated sodium channel 1.2-mediated current expressed in HEK293 cells at -60 to +10 mV holding poteinitial at 1 to 10 uM after 5 mins measured after drug washout by patch clamp electrophysiology | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
14. | ALA943771 | B | Inhibition of human Nav1.2 channel at 3 uM | Homo sapiens | 4 | single protein format | Scientific Literature | ||
15. | ALA943772 | B | Inhibition of human Nav1.2 channel at 1 uM | Homo sapiens | 4 | single protein format | Scientific Literature | ||
16. | ALA943773 | B | Inhibition of human Nav1.2 channel at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
17. | ALA943774 | B | Inhibition of human Nav1.2 channel at 0.1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
18. | ALA943775 | B | Inhibition of human Nav1.2 channel at 0.3 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
19. | ALA943776 | B | Inhibition of human Nav1.2 channel at 0.03 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
20. | ALA2155927 | B | Inhibition of human NaV1.2-mediated current at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature |