| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA921136 | B | Displacement of [3H]Ro15-1788 from GABAA alpha-1 receptor in Sprague-Dawley rat cerebellar membrane | Rattus norvegicus | 1 | ALA1143976 | assay format | Scientific Literature | |
| 2. | ALA921137 | B | Displacement of [3H]Ro15-1788 from GABAA alpha1 receptor in Sprague-Dawley rat cerebral cortex membrane | Rattus norvegicus | 1 | ALA1143976 | tissue-based format | Scientific Literature | |
| 3. | ALA979936 | B | Activity at rat wild type GABAA alpha-1-beta-2 receptor expressed in Xenopus laevis oocytes at -60 mV by Two-Electrode voltage clamp method | Rattus norvegicus | 1 | ALA1155944 | cell-based format | Scientific Literature | |
| 4. | ALA967929 | F | Agonist activity at rat wild type GABAA alpha-1-beta-2 receptor expressed in Xenopus laevis oocytes at -60 mV by Two-Electrode voltage clamp method | Rattus norvegicus | 1 | ALA1155944 | cell-based format | Scientific Literature | |
| 5. | ALA967932 | F | Agonist activity at rat wild type GABAA alpha-1-beta-2 receptor expressed in Xenopus laevis oocytes at -60 mV at 30 mM by Two-Electrode voltage clamp method | Rattus norvegicus | 1 | ALA1155944 | cell-based format | Scientific Literature | |
| 6. | ALA967935 | F | Agonist activity at rat wild type GABAA alpha-1-beta-2 receptor expressed in Xenopus laevis oocytes as inhibition of GABA-induced current at -60 mV by Two-Electrode voltage clamp method in presence of picrotoxinin | Rattus norvegicus | 1 | ALA1155944 | cell-based format | Scientific Literature | |
| 7. | ALA967938 | F | Agonist activity at rat wild type GABAA alpha-1-beta-2 receptor expressed in Xenopus laevis oocytes as inhibition of GABA-induced current at -60 mV at 1 mM by Two-Electrode voltage clamp method | Rattus norvegicus | 1 | ALA1155944 | cell-based format | Scientific Literature | |
| 8. | ALA971714 | F | Agonist activity at rat wild type GABAA alpha-1-beta-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of drug-induced current at -60 mV at 10 mM in presence of 100 uM picrotoxinin by Two-Electrode voltage clamp method | Rattus norvegicus | 1 | ALA1155944 | cell-based format | Scientific Literature | |
| 9. | ALA1031408 | B | Displacement of flunitrazepam from rat GABAA1 receptor at 3 uM | Rattus norvegicus | 1 | ALA1142492 | single protein format | Scientific Literature | |
| 10. | ALA1031409 | B | Displacement of muscimol from rat GABAA1 receptor at 3 uM | Rattus norvegicus | 1 | ALA1142492 | single protein format | Scientific Literature | |
| 11. | ALA3995200 | B | Displacement of [3H]RO15-1788 from recombinant rat GABAalpha1 receptor expressed in HEK293 cells after 1 hr | Rattus norvegicus | 3 | ALA3994587 | cell-based format | Scientific Literature | |
| 12. | ALA4219576 | B | Agonist activity at GABAA receptor in Sprague-Dawley rat forebrain membranes assessed as enhancement of [3H]muscimol binding after 2 hrs by radiometric analysis | Rattus norvegicus | 1 | ALA4219030 | assay format | Scientific Literature | |
| 13. | ALA4219577 | B | Agonist activity at GABAA receptor in Sprague-Dawley rat forebrain membranes assessed as enhancement of [3H]muscimol binding at 1 to 100 uM after 2 hrs by radiometric analysis relative to control | Rattus norvegicus | 1 | ALA4219030 | assay format | Scientific Literature | |
| 14. | ALA4881635 | B | BZD/CENTR/R Cerep selectivity data (BI) | Rattus norvegicus | 1 | ALA4507275 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 15. | ALA4881705 | B | BZD/CENTR/R Cerep selectivity data (BI) | Rattus norvegicus | 1 | ALA4507276 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 16. | ALA4881834 | B | GABAA MUSCIMOL CENT Eurofins-Panlabs selectivity data (BI) | Rattus norvegicus | 1 | ALA4507276 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 17. | ALA4881835 | B | GABAACENTR Eurofins-Panlabs selectivity data (BI) | Rattus norvegicus | 1 | ALA4507276 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 18. | ALA4882267 | B | GABAA MUSCIMOL CENT Eurofins-Panlabs selectivity data (BI) | Rattus norvegicus | 1 | ALA4507278 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 19. | ALA4882268 | B | GABAACENTR Eurofins-Panlabs selectivity data (BI) | Rattus norvegicus | 1 | ALA4507278 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 20. | ALA4882339 | B | GABAA MUSCIMOL CENT Eurofins-Panlabs selectivity data (BI) | Rattus norvegicus | 1 | ALA4507279 | single protein format | Donated Chemical Probes - SGC Frankfurt |
The page will load shortly, Thanks for your patience!