| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA686253 | F | Relative potency as ratio of the EC50 value of analogue to that of [PGlu6]SP6-11 in tachykinin receptor 3 in guinea pig ileum | Cavia porcellus | 2 | tissue-based format | Scientific Literature | ||
| 2. | ALA748091 | F | Effective dose was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methyl ester | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 3. | ALA748092 | F | Effective dose was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methyl ester. | Cavia porcellus | 2 | tissue-based format | Scientific Literature | ||
| 4. | ALA748093 | B | Evaluated for the binding affinity against NK3 receptor at 1 uM | Cavia porcellus | 1 | single protein format | Scientific Literature | ||
| 5. | ALA745028 | F | Compound was evaluated for NK-3 receptor antagonistic activity in the guinea pig trachea; Inactive | Cavia porcellus | 1 | assay format | Scientific Literature | ||
| 6. | ALA750064 | B | Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligand | Cavia porcellus | 3 | cell membrane format | Scientific Literature | ||
| 7. | ALA882643 | B | Inhibitory activity against binding of [125I][MePhe7]-NKB SP to tachykinin NK-3 receptor in guinea pig cortical membranes. | Cavia porcellus | 4 | cell membrane format | Scientific Literature | ||
| 8. | ALA872437 | B | NK3 IC50 determined using [125I]bolton Hunter labeled eledoisin at NK3 receptors from guinea pig cerebral cortex | Cavia porcellus | 3 | tissue-based format | Scientific Literature | ||
| 9. | ALA747335 | B | Inhibitory activity against binding of [125I][MePhe7]-NKB SP to tachykinin NK-3 receptor in guinea pig cortical membranes at concentration 10 uM | Cavia porcellus | 2 | cell membrane format | Scientific Literature | ||
| 10. | ALA857873 | B | The compound was tested for binding affinity against Tachykinin receptor 3 from guinea pig cerebral cortex | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 11. | ALA811320 | B | Ability to displace [3H]senktide succinyl-[Asp9MePhe8]-SP (6-13)} from Tachykinin receptor 3 of guinea pig cerebral cortex membrane | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 12. | ALA811321 | B | Binding affinity towards Tachykinin receptor 3 in guinea pig cerebral cortex using [3H]senktide as radioligand; Inactive (>>10 uM) | Cavia porcellus | 6 | tissue-based format | Scientific Literature | ||
| 13. | ALA811322 | B | Binding affinity towards Tachykinin receptor 3 in guinea pig cerebral cortex using [3H]senktide as radioligand; Value ranges from 5.8-14u M | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 14. | ALA811323 | B | Binding affinity towards Tachykinin receptor 3 in guinea pig cerebral cortex using [3H]senktide as radioligand; Value ranges from 8.2-9.4 uM | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 15. | ALA811324 | B | Compound was tested for binding affinity towards Tachykinin receptor 3 binding sites in guinea pig cortical membranes using [125I][MePhe7]-NKB as radioligand | Cavia porcellus | 1 | cell membrane format | Scientific Literature | ||
| 16. | ALA811325 | B | Compound was tested for binding affinity towards Tachykinin receptor 3 binding sites in guinea pig cortical membranes using [125I]-[MePhe7]-Neurokinin B as radioligand | Cavia porcellus | 1 | cell membrane format | Scientific Literature | ||
| 17. | ALA811326 | B | Concentration producing half-maximal inhibition of specific binding of [3H]senktide to Tachykinin receptor 3 in the guinea pig cerebral cortex | Cavia porcellus | 5 | tissue-based format | Scientific Literature | ||
| 18. | ALA811327 | B | Inhibitory activity against Tachykinin receptor 3 in guinea pig cortex [125I]-BH-eledoisin as radioligand | Cavia porcellus | 1 | assay format | Scientific Literature | ||
| 19. | ALA811328 | B | Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I]-[MePhe7] | Cavia porcellus | 3 | cell membrane format | Scientific Literature | ||
| 20. | ALA811329 | B | Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I][MePhe7]-NKB | Cavia porcellus | 2 | cell membrane format | Scientific Literature |
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