| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA655825 | B | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membrane compared to hCGRPalpha | Cavia porcellus | 9 | cell membrane format | Scientific Literature | ||
| 2. | ALA655826 | B | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation relative to hCGRPalpha. | Cavia porcellus | 9 | cell membrane format | Scientific Literature | ||
| 3. | ALA655827 | B | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation. | Cavia porcellus | 1 | cell membrane format | Scientific Literature | ||
| 4. | ALA655828 | B | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membrane | Cavia porcellus | 9 | cell membrane format | Scientific Literature | ||
| 5. | ALA655829 | B | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation | Cavia porcellus | 1 | cell membrane format | Scientific Literature | ||
| 6. | ALA654167 | B | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation. | Cavia porcellus | 7 | cell membrane format | Scientific Literature | ||
| 7. | ALA654168 | B | Compound was tested in vitro for its binding affinity towards recombinant human Calcitonin gene-related peptide type receptor (membranes of HEK293 cells) using [125I]hCGRP as radioligand | 1 | cell-based format | Scientific Literature | |||
| 8. | ALA654169 | B | Displacement of [125I]hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranes | Homo sapiens | 13 | assay format | Scientific Literature | ||
| 9. | ALA654170 | B | In vitro ability to displace [125 I]CGRP from Calcitonin gene-related peptide type receptor at 4 degrees Centigrade in rabbit lung | Oryctolagus cuniculus | 2 | single protein format | Scientific Literature | ||
| 10. | ALA654171 | B | In vitro ability to displace [125 I]CGRP from Calcitonin gene-related peptide type receptor at 4 degrees Celsius in rabbit lung; value ranges from (2-5) | Oryctolagus cuniculus | 1 | single protein format | Scientific Literature | ||
| 11. | ALA654172 | B | In vitro ability to displace [125 I]CGRP from Calcitonin gene-related peptide type receptor at 4 degrees Celsius in rabbit porcine c+i | Oryctolagus cuniculus | 3 | single protein format | Scientific Literature | ||
| 12. | ALA659129 | B | CGRP1 receptor affinity on human neuroblastoma cells SK-N-MC, which selectively express the human CGRP1 receptor. | 64 | assay format | Scientific Literature | |||
| 13. | ALA656585 | B | CGRP1 receptor affinity on human neuroblastoma cells SK-N-MC, which selectively express the human CGRP1 receptor. | 29 | assay format | Scientific Literature | |||
| 14. | ALA884938 | F | Antagonistic activity against calcitonin gene related peptide receptor determined by measuring the formation of cyclic AMP in SK-N-MC cells | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 15. | ALA884694 | B | Affinity against calcitonin gene related peptide receptor (1 uM) in marmoset tissue homogenates using [125I]CGRP as radioligand after 180 minutes of incubation at pH 7.40 | Callithrix | 2 | assay format | Scientific Literature | ||
| 16. | ALA884701 | B | Affinity against human calcitonin gene related peptide receptor (1 uM) expressed in SK-N-MC cells using [125I]-CGRP as radioligand after 180 minutes of incubation at pH 7.40 | Homo sapiens | 20 | cell-based format | Scientific Literature | ||
| 17. | ALA885294 | B | Affinity against calcitonin gene related peptide receptor (1 uM) in marmoset tissue homogenates using [125I]-CGRP as radioligand after 180 minutes of incubation at pH 7.40; n.d.=Not determined | Callithrix | 1 | assay format | Scientific Literature | ||
| 18. | ALA853349 | B | Inhibition of CGRP receptor at 1 uM | 1 | single protein format | Scientific Literature | |||
| 19. | ALA908626 | B | Displacement of [125I]CGRP from human recombinant CGRP receptor | Homo sapiens | 51 | single protein format | Scientific Literature | ||
| 20. | ALA908628 | F | Activity at CGRP receptor assessed as inhibition of CGRP-stimulated cAMP production | Homo sapiens | 36 | assay format | Scientific Literature |
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