# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA655825 | Binding | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membrane compared to hCGRPalpha | Cavia porcellus | 9 | ALA1126178 | cell membrane format | Scientific Literature | |
2. | ALA655826 | Binding | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation relative to hCGRPalpha. | Cavia porcellus | 9 | ALA1126178 | cell membrane format | Scientific Literature | |
3. | ALA655827 | Binding | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation. | Cavia porcellus | 1 | ALA1126178 | cell membrane format | Scientific Literature | |
4. | ALA655828 | Binding | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membrane | Cavia porcellus | 9 | ALA1126178 | cell membrane format | Scientific Literature | |
5. | ALA655829 | Binding | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation | Cavia porcellus | 1 | ALA1126178 | cell membrane format | Scientific Literature | |
6. | ALA654167 | Binding | Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane preparation. | Cavia porcellus | 7 | ALA1126178 | cell membrane format | Scientific Literature | |
7. | ALA654168 | Binding | Compound was tested in vitro for its binding affinity towards recombinant human Calcitonin gene-related peptide type receptor (membranes of HEK293 cells) using [125I]hCGRP as radioligand | 1 | ALA1150009 | cell-based format | Scientific Literature | ||
8. | ALA654169 | Binding | Displacement of [125I]hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranes | Homo sapiens | 13 | ALA1150009 | assay format | Scientific Literature | |
9. | ALA654170 | Binding | In vitro ability to displace [125 I]CGRP from Calcitonin gene-related peptide type receptor at 4 degrees Centigrade in rabbit lung | Oryctolagus cuniculus | 2 | ALA1128851 | single protein format | Scientific Literature | |
10. | ALA654171 | Binding | In vitro ability to displace [125 I]CGRP from Calcitonin gene-related peptide type receptor at 4 degrees Celsius in rabbit lung; value ranges from (2-5) | Oryctolagus cuniculus | 1 | ALA1128851 | single protein format | Scientific Literature | |
11. | ALA654172 | Binding | In vitro ability to displace [125 I]CGRP from Calcitonin gene-related peptide type receptor at 4 degrees Celsius in rabbit porcine c+i | Oryctolagus cuniculus | 3 | ALA1128851 | single protein format | Scientific Literature | |
12. | ALA659129 | Binding | CGRP1 receptor affinity on human neuroblastoma cells SK-N-MC, which selectively express the human CGRP1 receptor. | 64 | ALA1131198 | assay format | Scientific Literature | ||
13. | ALA656585 | Binding | CGRP1 receptor affinity on human neuroblastoma cells SK-N-MC, which selectively express the human CGRP1 receptor. | 29 | ALA1131198 | assay format | Scientific Literature | ||
14. | ALA1060867 | Binding | Displacement of [125I]human CGRP from human CLR expressed in HEK293 cells coexpressing human RAMP1 | Homo sapiens | 10 | ALA1153066 | cell-based format | Scientific Literature | |
15. | ALA1060868 | Functional | Antagonist activity at human CLR expressed in HEK293 cells coexpressing human RAMP1 assessed as inhibition of human CGRPalpha-induced cAMP production after 30 mins by scintillation proximity assay | Homo sapiens | 10 | ALA1153066 | cell-based format | Scientific Literature | |
16. | ALA1060869 | Functional | Antagonist activity at human CLR expressed in HEK293 cells coexpressing human RAMP1 assessed as inhibition of human CGRPalpha-induced cAMP production after 30 mins by scintillation proximity assay in presence of 50% human serum | Homo sapiens | 10 | ALA1153066 | cell-based format | Scientific Literature | |
17. | ALA1046104 | Binding | Displacement of [125I]human CGRP from human CLR expressed in HEK 293 cells coexpressing human RAMP1 after 3 hrs by scintillation counting | Homo sapiens | 21 | ALA1156095 | cell-based format | Scientific Literature | |
18. | ALA1046105 | Functional | Antagonist activity at human CLR expressed in HEK293 cells coexpressing human RAMP1 assessed as inhibition of human CGRPalpha-induced cAMP production after 5 mins by scintillation proximity assay | Homo sapiens | 11 | ALA1156095 | cell-based format | Scientific Literature | |
19. | ALA1046106 | Functional | Antagonist activity at human CLR expressed in HEK293 cells coexpressing human RAMP1 assessed as inhibition of human CGRPalpha-induced cAMP production after 5 mins in presence of 50% human serum by scintillation proximity assay | Homo sapiens | 11 | ALA1156095 | cell-based format | Scientific Literature | |
20. | ALA1050773 | Binding | Displacement of [125I]hCGRP from human cloned CGRP receptor expressed in HEK293 cells | Homo sapiens | 18 | ALA1156010 | cell-based format | Scientific Literature |