# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1062777 | Binding | Binding constant for GAK kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1062807 | Binding | Percentage GAK activity remaining in the presence of 10uM inhibitor | Homo sapiens | 4 | ALA1150976 | single protein format | Scientific Literature | |
3. | ALA1062013 | Binding | Percentage GAK activity remaining in the presence of 1uM inhibitor | Homo sapiens | 9 | ALA1150976 | single protein format | Scientific Literature | |
4. | ALA1049978 | Binding | Binding affinity to GAK assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | ALA1154183 | single protein format | Scientific Literature | ||
5. | ALA1053743 | Binding | Inhibition of GAK assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
6. | ALA988955 | Binding | Binding affinity to human GAK | Homo sapiens | 1 | ALA1151712 | single protein format | Scientific Literature | |
7. | ALA993455 | Binding | Binding affinity to human GAK at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
8. | ALA1004484 | Binding | Binding affinity to human recombinant GAK expressed in Escherichia coli assessed as thermal shift by differential scanning fluorimetry | Homo sapiens | 7 | ALA1140872 | assay format | Scientific Literature | |
9. | ALA974029 | Binding | Inhibition of Gak | 2 | ALA1149823 | single protein format | Scientific Literature | ||
10. | ALA984521 | Binding | Inhibition of GAK at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
11. | ALA831128 | Binding | Inhibition of human cyclin G associated kinase at 100 uM ATP | Homo sapiens | 1 | ALA1139545 | single protein format | Scientific Literature | |
12. | ALA860789 | Binding | Average Binding Constant for GAK; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
13. | ALA862341 | Binding | Inhibition of GAK at 10 uM | Homo sapiens | 1 | ALA1138177 | single protein format | Scientific Literature | |
14. | ALA1169247 | Binding | Inhibition of GAK at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
15. | ALA1174438 | Binding | Inhibition of GAK at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
16. | ALA1244370 | Binding | Inhibition of GAK | 1 | ALA1240341 | single protein format | Scientific Literature | ||
17. | ALA1244854 | Binding | Binding affinity to GAK | 7 | ALA1240346 | single protein format | Scientific Literature | ||
18. | ALA1259874 | Binding | Inhibition of GAK at 10 uM relative to control | 1 | ALA1255531 | single protein format | Scientific Literature | ||
19. | ALA1769110 | Binding | Inhibition of GAK at 10 uM | 2 | ALA1764984 | single protein format | Scientific Literature | ||
20. | ALA1769122 | Binding | Inhibition of GAK | 2 | ALA1764984 | single protein format | Scientific Literature |