| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA830019 | B | Inhibition of human receptor-interacting serine-threonine kinase 2 (RIPK2) at 100 uM ATP | Homo sapiens | 1 | ALA1139545 | single protein format | Scientific Literature | |
| 2. | ALA860788 | B | Average Binding Constant for RIPK2; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
| 3. | ALA922158 | B | Activity of human RIPK2 kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
| 4. | ALA975465 | B | Inhibition of human RIPK2 kinase assessed as residual enzyme activity at 0.1 uM | Homo sapiens | 1 | ALA1155876 | single protein format | Scientific Literature | |
| 5. | ALA995020 | B | Inhibition of RIPK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 6. | ALA1025751 | B | Binding affinity to human RIPK2 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
| 7. | ALA1055110 | B | Inhibition of RIPK2 at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
| 8. | ALA1052973 | B | Percentage RIP2 activity remaining in the presence of 10uM inhibitor | Homo sapiens | 4 | ALA1150976 | single protein format | Scientific Literature | |
| 9. | ALA1062023 | B | Percentage RIP2 activity remaining in the presence of 1uM inhibitor | Homo sapiens | 9 | ALA1150976 | single protein format | Scientific Literature | |
| 10. | ALA1051312 | B | Binding constant for RIPK2 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 11. | ALA1051329 | B | Inhibition of RIP2 in the presence of 100uM ATP | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
| 12. | ALA1043886 | B | Binding affinity to RIPK2 assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | ALA1154183 | single protein format | Scientific Literature | ||
| 13. | ALA1052948 | B | Inhibition of RIPK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 14. | ALA1043797 | B | Residual activity of RIPK2 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 15. | ALA1072504 | B | Residual activity of RIPK2 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 16. | ALA1071357 | B | Residual activity of RIPK2 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 17. | ALA1108059 | B | Inhibition of RIPK2 at 10 uM assessed as residual activity by [33P]ATP radioactive filter binding assay relative to control | 2 | ALA1156950 | single protein format | Scientific Literature | ||
| 18. | ALA1166844 | B | Inhibition of RIPK2 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
| 19. | ALA1175254 | B | Inhibition of RIPK2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 20. | ALA1221006 | B | Inhibition of human RIP2 autophosphorylation expressed in HEK293T cells | Homo sapiens | 2 | ALA1212703 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!