# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA834935 | F | In vitro inhibition of Na-dependent [14C]AMG uptake in CHO-K1 cells expressing human sodium glucose co-transporter 2 | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
2. | ALA863286 | B | Inhibitory activity towards human SGLT2 expressed in CHO-K1 cells | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
3. | ALA863288 | B | Inhibitory activity towards human SGLT2 expressed in CHO-K1 cells at 10 uM | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
4. | ALA869552 | B | Inhibitory activity against SGLT2 expressed in CHO-K1 cells | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
5. | ALA868398 | B | Inhibition of SGLT2 expressed in CHO-K1 cells at 10 uM | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
6. | ALA1811698 | B | Inhibition of human SGLT2 expressed in african green monkey COS7 cells assessed as inhibition of [14C]-methyl-alpha-D-glucopyranoside uptake after 2 hrs by scintillation counting in presence of 25 % human plasma | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
7. | ALA1811701 | B | Inhibition of human SGLT2 expressed in human 293 cells assessed as inhibition of [14C]-methyl-alpha-D-glucopyranoside uptake at 10 nM after 1.5 hrs by scintillation counting in presence of 25 % human plasma | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
8. | ALA892511 | B | Inhibition of human SGLT2 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake at 50 uM | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
9. | ALA892513 | B | Inhibition of human SGLT2 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
10. | ALA1680964 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-alpha-methyl-D-glucopyranoside uptake after 2 hrs by liquid scintillation counting | Homo sapiens | 47 | cell-based format | Scientific Literature | ||
11. | ALA2021179 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation counting | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
12. | ALA1821091 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as reduction of [14C]-labeled AMG after 2 hrs by liquid scintillation counting | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
13. | ALA2051076 | B | Inhibition of human SGLT2 expressed in CHO-K1 cells by [14C]AMG uptake assay | Homo sapiens | 18 | cell-based format | Scientific Literature | ||
14. | ALA2065401 | B | Inhibition of human SGLT2 expressed in CHO-K1 cells incubated for 120 mins at 37 degC by [14C]-AMG uptake assay | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
15. | ALA1788054 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-alpha-methyl-D-glucopyranoside uptake after 2 hrs by liquid scintillation counter | Homo sapiens | 45 | cell-based format | Scientific Literature | ||
16. | ALA947997 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as inhibition of [14C]AMG accumulation | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
17. | ALA1005353 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]alpha-methyl-D-glucopyranoside uptake by fluorescence polarization assay | Homo sapiens | 32 | cell-based format | Scientific Literature | ||
18. | ALA977366 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as intracellular accumulation of [14C]alpha-methyl glucopyranoside | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
19. | ALA977369 | B | Inhibition of human SGLT2 expressed in Xenopus oocyte assessed as [14C]alpha-methyl glucopyranoside uptake | Homo sapiens | 2 | assay format | Scientific Literature | ||
20. | ALA961709 | B | Inhibition of human kidney SGLT2 assessed as renal glucose reabsorption | Homo sapiens | 8 | single protein format | Scientific Literature |