# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA834935 | F | In vitro inhibition of Na-dependent [14C]AMG uptake in CHO-K1 cells expressing human sodium glucose co-transporter 2 | Homo sapiens | 23 | ALA1137899 | cell-based format | Scientific Literature | |
2. | ALA863286 | B | Inhibitory activity towards human SGLT2 expressed in CHO-K1 cells | Homo sapiens | 11 | ALA1141232 | cell-based format | Scientific Literature | |
3. | ALA863288 | B | Inhibitory activity towards human SGLT2 expressed in CHO-K1 cells at 10 uM | Homo sapiens | 2 | ALA1141232 | cell-based format | Scientific Literature | |
4. | ALA869552 | B | Inhibitory activity against SGLT2 expressed in CHO-K1 cells | Homo sapiens | 22 | ALA1139015 | cell-based format | Scientific Literature | |
5. | ALA868398 | B | Inhibition of SGLT2 expressed in CHO-K1 cells at 10 uM | Homo sapiens | 5 | ALA1139015 | cell-based format | Scientific Literature | |
6. | ALA892511 | B | Inhibition of human SGLT2 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake at 50 uM | Homo sapiens | 9 | ALA1147913 | cell-based format | Scientific Literature | |
7. | ALA892513 | B | Inhibition of human SGLT2 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake | Homo sapiens | 3 | ALA1147913 | cell-based format | Scientific Literature | |
8. | ALA947997 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as inhibition of [14C]AMG accumulation | Homo sapiens | 5 | ALA1142359 | cell-based format | Scientific Literature | |
9. | ALA1005353 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]alpha-methyl-D-glucopyranoside uptake by fluorescence polarization assay | Homo sapiens | 32 | ALA1141694 | cell-based format | Scientific Literature | |
10. | ALA977366 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as intracellular accumulation of [14C]alpha-methyl glucopyranoside | Homo sapiens | 16 | ALA1140039 | cell-based format | Scientific Literature | |
11. | ALA977369 | B | Inhibition of human SGLT2 expressed in Xenopus oocyte assessed as [14C]alpha-methyl glucopyranoside uptake | Homo sapiens | 2 | ALA1140039 | assay format | Scientific Literature | |
12. | ALA961709 | B | Inhibition of human kidney SGLT2 assessed as renal glucose reabsorption | Homo sapiens | 8 | ALA1153320 | single protein format | Scientific Literature | |
13. | ALA1043168 | B | Inhibition of human SGLT2 expressed in HEK293.ETN cells assessed as methyl-alpha-D-[U-14C]glucopyranoside uptake by scintillation counting | Homo sapiens | 3 | ALA1155186 | cell-based format | Scientific Literature | |
14. | ALA1043169 | B | Inhibition of human SGLT2 expressed in HEK293.ETN cells assessed as methyl-alpha-D-[U-14C]glucopyranoside uptake at 1 uM by scintillation counting | Homo sapiens | 1 | ALA1155186 | cell-based format | Scientific Literature | |
15. | ALA1043173 | B | Inhibition of human SGLT2 expressed in HEK293.ETN cells assessed as methyl-alpha-D-[U-14C]glucopyranoside uptake at 10 nM by scintillation counting | Homo sapiens | 1 | ALA1155186 | cell-based format | Scientific Literature | |
16. | ALA1040741 | B | Inhibition of human SGLT2 expressed in HEK293 cells assessed as inhibition of [14C]alpha-methylglucopyranoside uptake | Homo sapiens | 23 | ALA1156071 | cell-based format | Scientific Literature | |
17. | ALA1050643 | B | Inhibition of human SGLT2 transfected in HEK293.ETN cells assessed as AMG uptake after 1.5 hrs by scintillation counting | Homo sapiens | 27 | ALA1156745 | cell-based format | Scientific Literature | |
18. | ALA1068133 | B | Inhibition of human SGLT2 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake at 50 uM | Homo sapiens | 20 | ALA1159054 | cell-based format | Scientific Literature | |
19. | ALA1068136 | B | Inhibition of human SGLT2 expressed in COS1 cells assessed as [14C]methyl-alpha-D-glucopyranoside uptake at 0.2 uM | Homo sapiens | 1 | ALA1159054 | cell-based format | Scientific Literature | |
20. | ALA1070174 | B | Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation counting | Homo sapiens | 14 | ALA1157651 | cell-based format | Scientific Literature |