| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA680343 | F | Effective dose by H3-mediated bronchospasm in guinea pig | Cavia porcellus | 2 | tissue-based format | Scientific Literature | ||
| 2. | ALA680344 | B | In vitro effective concentration for H-3-mediated contraction of guinea pig ileum | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 3. | ALA680345 | F | In vitro effective concentration for H-3-mediated contraction of guinea pig ileum | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 4. | ALA683997 | F | Evaluated in vivo for its H3 receptor antagonist activity in the CNS hypertension model | Cavia porcellus | 6 | organism-based format | Scientific Literature | ||
| 5. | ALA688090 | F | Evaluated in vivo for its H3 receptor antagonist activity in the CNS hypertension model at 3 mg/kg dose | Cavia porcellus | 5 | organism-based format | Scientific Literature | ||
| 6. | ALA689677 | F | H3 -antagonist potency determined in electrically stimulated guinea-pig ileum | Cavia porcellus | 19 | tissue-based format | Scientific Literature | ||
| 7. | ALA686856 | F | Inhibition of H3-receptor mediated neurogenic contractions in the isolated guinea pig ileum assay | Cavia porcellus | 12 | tissue-based format | Scientific Literature | ||
| 8. | ALA687404 | F | Compound was tested for inhibition of histamine H3-receptor mediated neurogenic contractions in the isolated guinea pig ileum assay; Partial agonist | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 9. | ALA687982 | F | Compound was tested for inhibition of histamine H3-receptor mediated neurogenic contractions in the isolated guinea pig ileum assay; Full agonist | Cavia porcellus | 3 | tissue-based format | Scientific Literature | ||
| 10. | ALA693933 | F | Tested for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of 1-3 micro M, not determined | Cavia porcellus | 1 | assay format | Scientific Literature | ||
| 11. | ALA693934 | F | Tested for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of 1-3 micro M; not determined | Cavia porcellus | 4 | assay format | Scientific Literature | ||
| 12. | ALA693935 | F | Compound was tested in vitro against histamine H3 receptor mediated inhibition of cholinergic neurogenic contractions in isolated guinea pig ileum; Not tested | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 13. | ALA693936 | F | Compound was tested for the agonist activity against histamine H3 receptor of guinea pig ileum; ND = Not determined | Cavia porcellus | 1 | tissue-based format | Scientific Literature | ||
| 14. | ALA693937 | B | Compound was evaluated for its inhibitory activity against Histamine H3 receptor of guinea pig brain membrane at a concentration of 1 ug/mL | Cavia porcellus | 2 | assay format | Scientific Literature | ||
| 15. | ALA693938 | B | Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptors in homogenates of rat cerebral cortex | Cavia porcellus | 11 | tissue-based format | Scientific Literature | ||
| 16. | ALA693939 | B | Activity at Histamine H3 receptor using functional H3 receptor assay on guinea pig ileum | Cavia porcellus | 9 | tissue-based format | Scientific Literature | ||
| 17. | ALA693940 | F | Compound was evaluated for its antagonist affinity towards Histamine H3 receptor of guinea pig | Cavia porcellus | 5 | assay format | Scientific Literature | ||
| 18. | ALA693941 | F | Histamine H3-antagonist potency on electrically stimulated guinea pig ileum | Cavia porcellus | 10 | tissue-based format | Scientific Literature | ||
| 19. | ALA693942 | F | Compound was tested for H3-antagonist potency on electrically stimulated guinea pig ileum; Unsurmountable antagonism at concentration > 10-7 M | Cavia porcellus | 2 | tissue-based format | Scientific Literature | ||
| 20. | ALA693943 | F | Compound was tested for the agonist activity against histamine H3 receptor of guinea pig ileum | Cavia porcellus | 7 | tissue-based format | Scientific Literature |
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