| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA676728 | B | Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A); d indicates Not determined | Oryctolagus cuniculus | 1 | ALA1127771 | assay format | Scientific Literature | |
| 2. | ALA677396 | B | Binding affinity against endothelin A receptor from rabbit renal vascular smooth muscles | Oryctolagus cuniculus | 52 | ALA1128478 | single protein format | Scientific Literature | |
| 3. | ALA679789 | B | Compound was evaluated for binding affinity against rabbit Endothelin A receptor | Oryctolagus cuniculus | 1 | ALA1129233 | single protein format | Scientific Literature | |
| 4. | ALA679790 | B | Compound was evaluated for the receptor binding activity in rabbit artery vascular smooth muscle cells expressing Endothelin A receptor | Oryctolagus cuniculus | 3 | ALA1129097 | tissue-based format | Scientific Literature | |
| 5. | ALA679791 | F | Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells. | Oryctolagus cuniculus | 28 | ALA1128950 | tissue-based format | Scientific Literature | |
| 6. | ALA679792 | F | Compound was tested for inhibition of binding of [125I]ET1 to cloned human Endothelin A receptor expressed in LtK- cells | Oryctolagus cuniculus | 1 | ALA1128950 | cell-based format | Scientific Literature | |
| 7. | ALA679793 | F | Compound was tested for its ability to inhibit Endothelin A receptor induced arachidonic acid release(AARA) in rabbit renal artery vascular smooth muscles. | Oryctolagus cuniculus | 4 | ALA1128950 | tissue-based format | Scientific Literature | |
| 8. | ALA679794 | B | Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cells | Oryctolagus cuniculus | 13 | ALA1127199 | assay format | Scientific Literature | |
| 9. | ALA679795 | B | Inhibition of ET-1 binding to Endothelin A receptor in cultured rabbit renal artery vascular smooth muscle cells | Oryctolagus cuniculus | 10 | ALA1126242 | assay format | Scientific Literature | |
| 10. | ALA679796 | F | Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cells | Oryctolagus cuniculus | 28 | ALA1128478 | assay format | Scientific Literature | |
| 11. | ALA679797 | B | Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cells | Oryctolagus cuniculus | 9 | ALA1129982 | assay format | Scientific Literature | |
| 12. | ALA679798 | B | Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cells | Oryctolagus cuniculus | 14 | ALA1159137 | assay format | Scientific Literature | |
| 13. | ALA679799 | B | Inhibition of binding to Endothelin A receptor of rabbit renal vascular smooth muscle cells | Oryctolagus cuniculus | 14 | ALA1130387 | assay format | Scientific Literature | |
| 14. | ALA873588 | F | Tested for antagonistic activity against Endothelin A receptor in the rabbit renal artery vascular smooth muscle cells. | Oryctolagus cuniculus | 15 | ALA1128292 | assay format | Scientific Literature | |
| 15. | ALA676566 | B | Tested for binding affinity towards rabbit Endothelin A receptor | Oryctolagus cuniculus | 3 | ALA1133352 | single protein format | Scientific Literature | |
| 16. | ALA676567 | B | The inhibitory constant was evaluated against Endothelin A receptor in rabbit renal artery tissue | Oryctolagus cuniculus | 1 | ALA1127202 | single protein format | Scientific Literature | |
| 17. | ALA676568 | F | Antagonism of ET-1 induced increase in intracellular Ca+2 in rabbit carotid artery rings | Oryctolagus cuniculus | 8 | ALA1127313 | tissue-based format | Scientific Literature | |
| 18. | ALA676569 | B | Ability to inhibit Endothelin A receptor induced contractions in rabbit carotid artery rings (ETA) was determined in an in vitro functional assay. | Oryctolagus cuniculus | 42 | ALA1131435 | tissue-based format | Scientific Literature | |
| 19. | ALA676570 | B | Ability to inhibit Endothelin A receptor induced contractions in rabbit carotid artery rings (ETA) was determined in an in vitro functional assay. | Oryctolagus cuniculus | 15 | ALA1131435 | tissue-based format | Scientific Literature | |
| 20. | ALA676571 | B | Inhibition of ET-1 induced contraction of rabbit femoral artery rings (Endothelin A receptor mediated) | Oryctolagus cuniculus | 9 | ALA1129982 | tissue-based format | Scientific Literature |
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