| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA810064 | B | Inhibitory activity against TRH using [3H]TRH at 10e-5 (M) | 1 | single protein format | Scientific Literature | |||
| 2. | ALA917826 | B | Displacement of [3H]N(1)-Me-His-TRH from TRHR1 | 18 | single protein format | Scientific Literature | |||
| 3. | ALA917828 | F | Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activity | 18 | cell-based format | Scientific Literature | |||
| 4. | ALA1809429 | B | Inhibition of Thyrotropin releasing hormone receptor at 4 uM | 1 | single protein format | Scientific Literature | |||
| 5. | ALA931825 | B | Inhibition of TRH receptor | 1 | single protein format | Scientific Literature | |||
| 6. | ALA1737857 | F | PUBCHEM_BIOASSAY: qHTS for Small Molecule Agonists and Allosteric Enhancers of Human TRH Receptor: Confirmation Screen for Enhancers. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID485365] | Homo sapiens | 69 | assay format | PubChem BioAssays | ||
| 7. | ALA1737990 | F | PUBCHEM_BIOASSAY: qHTS for Small Molecule Agonists and Allosteric Enhancers of Human TRH Receptor: Confirmation Screen for Agonists. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID485365, AID493056] | Homo sapiens | 197 | assay format | PubChem BioAssays | ||
| 8. | ALA2213034 | B | Inhibition of TRH receptor at 10 uM by CEREP assay | 1 | single protein format | Scientific Literature | |||
| 9. | ALA2388540 | B | Inhibition of human TRH1 receptor at 10 uM relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 10. | ALA3777183 | B | Binding affinity to human TRH1 receptor at 10 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4311080 | B | Displacement of [3H]Me-TRH from human recombinant TRH receptor at 10 uM after 120 mins by scintillation counting analysis relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 12. | ALA4358665 | B | Activity at human TRH receptor up to 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4882985 | B | Thyrotropin Releasing Hormone (TRH) Eurofins-Panlabs radioligand binding assay | Rattus | 4 | single protein format | Donated Chemical Probes - SGC Frankfurt | ||
| 14. | ALA5034717 | B | Displacement of [3H]Me-TRH from human recombinant TRH receptor at 10 uM after 120 mins by scintillation counting analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature |
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