# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860785 | B | Average Binding Constant for MARK2; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
2. | ALA860207 | B | Inhibition of EMK | Homo sapiens | 6 | ALA1148638 | single protein format | Scientific Literature | |
3. | ALA867307 | B | Inhibition of EMK | Homo sapiens | 1 | ALA1138045 | single protein format | Scientific Literature | |
4. | ALA913850 | B | Inhibition of EMK | Homo sapiens | 3 | ALA1142994 | single protein format | Scientific Literature | |
5. | ALA891247 | B | Inhibition of EMK by radiometric assay | Homo sapiens | 2 | ALA1147174 | single protein format | Scientific Literature | |
6. | ALA894156 | B | Inhibition of recombinant EMK by radiometric assay | Homo sapiens | 2 | ALA1148724 | single protein format | Scientific Literature | |
7. | ALA942723 | B | Inhibition of EMK | 1 | ALA1140564 | single protein format | Scientific Literature | ||
8. | ALA922022 | B | Activity of human PAR1Balpha kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
9. | ALA975455 | B | Inhibition of human PAR-1Balpha kinase assessed as residual enzyme activity at 0.1 uM | Homo sapiens | 1 | ALA1155876 | single protein format | Scientific Literature | |
10. | ALA987180 | B | Inhibition of MARK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
11. | ALA982752 | B | Binding affinity to human MARK2 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
12. | ALA1057488 | B | Inhibition of PAR-1Balpha at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
13. | ALA1049903 | B | Binding constant for MARK2 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
14. | ALA1049123 | B | Inhibition of MARK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
15. | ALA1041398 | B | Inhibition of PAR-1Balpha at 1 uM | 1 | ALA1154622 | single protein format | Scientific Literature | ||
16. | ALA1044530 | B | Inhibition of human MARK2 at 20 uM by FRET assay | Homo sapiens | 1 | ALA1156108 | single protein format | Scientific Literature | |
17. | ALA1040682 | B | Residual activity of MARK2 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
18. | ALA1041140 | B | Residual activity of MARK2 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
19. | ALA1050293 | B | Residual activity of MARK2 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
20. | ALA1100960 | B | Inhibition of MARK2 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature |