# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860782 | B | Average Binding Constant for STK17B; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
2. | ALA990545 | B | Inhibition of STK17b | 1 | ALA1149823 | single protein format | Scientific Literature | ||
3. | ALA986221 | B | Binding affinity to human DRAK2 | Homo sapiens | 1 | ALA1151712 | single protein format | Scientific Literature | |
4. | ALA982770 | B | Binding affinity to human DRAK2 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
5. | ALA1034105 | B | Inhibition of DRAK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
6. | ALA1060189 | B | Binding constant for full-length DRAK2 | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
7. | ALA1055296 | B | Inhibition of DRAK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
8. | ALA1168859 | B | Inhibition of DRAK2 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
9. | ALA1174321 | B | Inhibition of DRAK2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
10. | ALA1244797 | B | Binding affinity to DRAK2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
11. | ALA1646187 | B | Inhibition of human DYRK2 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
12. | ALA1826919 | B | Activity of DRAK2 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
13. | ALA1908639 | B | Binding constant for DRAK2 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
14. | ALA1947292 | B | Binding affinity to DRAK2 assessed as change in thermal denaturation at 10 uM by thermal stability shift assay | 17 | ALA1944596 | single protein format | Scientific Literature | ||
15. | ALA1959402 | B | Inhibition of STK17B at 1 uM | 1 | ALA1955770 | single protein format | Scientific Literature | ||
16. | ALA2214450 | B | Inhibition of STK17B | 1 | ALA2203257 | single protein format | Scientific Literature | ||
17. | ALA2216436 | B | Inhibition of DRAK2 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
18. | ALA2428155 | B | Competitive binding affinity to DRAK2 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
19. | ALA2429304 | B | Competitive binding affinity to STK17B (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | ALA2424622 | single protein format | Scientific Literature | |
20. | ALA3101918 | B | Inhibition of human DYRK2 assessed as residual activity at 1 uM relative to control | Homo sapiens | 1 | ALA3098105 | single protein format | Scientific Literature |