# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860782 | B | Average Binding Constant for STK17B; NA=Not Active at 10 uM | Homo sapiens | 20 | single protein format | Scientific Literature | ||
2. | ALA1826919 | B | Activity of DRAK2 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
3. | ALA1908639 | B | Binding constant for DRAK2 kinase domain | 72 | single protein format | Scientific Literature | |||
4. | ALA1947292 | B | Binding affinity to DRAK2 assessed as change in thermal denaturation at 10 uM by thermal stability shift assay | 17 | single protein format | Scientific Literature | |||
5. | ALA1959402 | B | Inhibition of STK17B at 1 uM | 1 | single protein format | Scientific Literature | |||
6. | ALA990545 | B | Inhibition of STK17b | 1 | single protein format | Scientific Literature | |||
7. | ALA986221 | B | Binding affinity to human DRAK2 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA982770 | B | Binding affinity to human DRAK2 at 10 uM relative to control | Homo sapiens | 17 | single protein format | Scientific Literature | ||
9. | ALA1034105 | B | Inhibition of DRAK2 at 3 uM | 1 | single protein format | Scientific Literature | |||
10. | ALA1060189 | B | Binding constant for full-length DRAK2 | Homo sapiens | 38 | single protein format | Scientific Literature | ||
11. | ALA1055296 | B | Inhibition of DRAK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
12. | ALA1168859 | B | Inhibition of DRAK2 at 1 uM | 6 | single protein format | Scientific Literature | |||
13. | ALA1174321 | B | Inhibition of DRAK2 at 10 uM | 2 | single protein format | Scientific Literature | |||
14. | ALA1244797 | B | Binding affinity to DRAK2 | 7 | single protein format | Scientific Literature | |||
15. | ALA1646187 | B | Inhibition of human DYRK2 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
16. | ALA2214450 | B | Inhibition of STK17B | 1 | single protein format | Scientific Literature | |||
17. | ALA2216436 | B | Inhibition of DRAK2 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
18. | ALA2428155 | B | Competitive binding affinity to DRAK2 (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
19. | ALA2429304 | B | Competitive binding affinity to STK17B (unknown origin) at 10 uM in presence of ATP relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
20. | ALA5256607 | B | Inhibition of wild type human DRAK2 at 1 uM by DiscoverX scanMAX assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature |