# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860776 | B | Average Binding Constant for TTK; NA=Not Active at 10 uM | Homo sapiens | 20 | single protein format | Scientific Literature | ||
2. | ALA2044153 | B | Inhibition of MPS1 by caliper method | 4 | single protein format | Scientific Literature | |||
3. | ALA2044939 | B | Inhibition of TTK at 1 uM | 1 | single protein format | Scientific Literature | |||
4. | ALA2044940 | B | Inhibition of TTK at 0.1 uM | 1 | single protein format | Scientific Literature | |||
5. | ALA2049463 | B | Inhibition of N-terminus FLAG-tagged TTK expressed in baculovirus expression system using [gamma-33P]-ATP measured after 60 mins by scintillation counting | 1 | assay format | Scientific Literature | |||
6. | ALA2049891 | B | Inhibition of Mps1 | 36 | single protein format | Scientific Literature | |||
7. | ALA1809661 | B | Inhibition of MPS1 assessed as [33P]-gamma-ATP incorporation into substrate P38-betatide by gamma counting | 25 | single protein format | Scientific Literature | |||
8. | ALA1826907 | B | Activity of TTK kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
9. | ALA1826262 | B | Inhibition of TTK assessed as residual activity at 10 uM by radioactivity assay in presence of 20 uM ATP | 1 | single protein format | Scientific Literature | |||
10. | ALA1908607 | B | Binding constant for TTK kinase domain | 72 | single protein format | Scientific Literature | |||
11. | ALA1925204 | B | Inhibition of N-terminus flag-tagged TTK expressed in baculovirus infected insect cells using [gamma33P]ATP as substrate after 60 mins by scintillation counting | 1 | cell-based format | Scientific Literature | |||
12. | ALA1930475 | B | Inhibition of TTK assessed as residual activity at 10 uM using [33P-ATP] by radiometric filter binding assay | 1 | single protein format | Scientific Literature | |||
13. | ALA1959410 | B | Inhibition of TTK at 1 uM | 1 | single protein format | Scientific Literature | |||
14. | ALA1664104 | B | Inhibition of TTK at 1 uM | 2 | single protein format | Scientific Literature | |||
15. | ALA2015824 | B | Inhibition of TTK assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
16. | ALA2014715 | B | Inhibition of TTK assessed as residual activity at 1 uM relative to control | 1 | single protein format | Scientific Literature | |||
17. | ALA2015526 | B | Inhibition of TTK at 10 uM | 1 | single protein format | Scientific Literature | |||
18. | ALA1962098 | B | GSK_PKIS: TTK mean inhibition at 0.1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
19. | ALA1962193 | B | GSK_PKIS: TTK mean inhibition at 1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
20. | ALA2150269 | B | Inhibition of N-terminal FLAG-tagged TTK expressed in baculovirus after 5 mins by scintillation counter | 1 | assay format | Scientific Literature |