# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860774 | B | Average Binding Constant for CLK1; NA=Not Active at 10 uM | Homo sapiens | 20 | single protein format | Scientific Literature | ||
2. | ALA1805398 | B | Inhibition of CLK1 transfected in human HeLa cells assessed as increase in exon inclusion ratio after 24 hrs by RT-PCR analysis | 4 | cell-based format | Scientific Literature | |||
3. | ALA1804240 | B | Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrate | Homo sapiens | 36 | single protein format | Scientific Literature | ||
4. | ALA898067 | B | Inhibition of CLK at 1 uM | 1 | single protein format | Scientific Literature | |||
5. | ALA2073010 | B | Inhibition of CLK1 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
6. | ALA1794519 | B | PUBCHEM_BIOASSAY: MLPCN Dyrk1A - CLK1 Selectivity Assay Measured in Biochemical System Using Plate Reader - 2124-05_Inhibitor_Dose_CherryPick_Activity. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504442] | 155 | biochemical format | PubChem BioAssays | |||
7. | ALA2014910 | B | Inhibition of CLK1 at 10 uM | 1 | single protein format | Scientific Literature | |||
8. | ALA1805117 | B | Inhibition of recombinant CLK1-mediated SR 9G8 protein phosphorylation at 10 uM after 30 mins by SDS-PAGE followed by autoradiography | 1 | single protein format | Scientific Literature | |||
9. | ALA1805120 | B | Inhibition of CLK1-mediated SRp55 protein phosphorylation in TNFalpha-stimulated human HMEC1 cells after 1 hr by Western blot analysis | 1 | cell-based format | Scientific Literature | |||
10. | ALA1805394 | B | Inhibition of CLK1-mediated SRp75 protein phosphorylation in TNFalpha-stimulated human HMEC1 cells after 1 hr by Western blot analysis | 1 | cell-based format | Scientific Literature | |||
11. | ALA1827761 | B | Activity of CLK1 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
12. | ALA1787822 | B | Inhibition of CLK1 at 10 uM | 1 | single protein format | Scientific Literature | |||
13. | ALA949031 | B | Inhibition of CLK1 | 1 | single protein format | Scientific Literature | |||
14. | ALA970578 | B | Inhibition of CLK1 at 1 uM | 1 | single protein format | Scientific Literature | |||
15. | ALA989739 | B | Inhibition of CLK1 | 1 | single protein format | Scientific Literature | |||
16. | ALA983555 | B | Binding affinity to human CLK1 at 10 uM relative to control | Homo sapiens | 17 | single protein format | Scientific Literature | ||
17. | ALA1032273 | B | Inhibition of CLK1 at 3 uM | 1 | single protein format | Scientific Literature | |||
18. | ALA963875 | B | Binding affinity to CLK1 | 4 | single protein format | Scientific Literature | |||
19. | ALA960117 | B | Inhibition of CLK1 | 1 | single protein format | Scientific Literature | |||
20. | ALA1050838 | B | Binding constant for full-length CLK1 | Homo sapiens | 38 | single protein format | Scientific Literature |