# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3430842 | Binding | Delta TM value showing the stabilisation of MST1 produced by compound binding | Homo sapiens | 156 | ALA1145498 | single protein format | Scientific Literature | |
2. | ALA3595431 | Binding | Inhibition of recombinant human MST1 at 1 uM relative to control | Homo sapiens | 1 | ALA3593241 | single protein format | Scientific Literature | |
3. | ALA3631456 | Binding | Inhibition of MST1 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
4. | ALA3739151 | Binding | Inhibition of MST1 (unknown origin) at 200 nM by electrophoretic mobility shift assay | Homo sapiens | 2 | ALA3734671 | single protein format | Scientific Literature | |
5. | ALA3751270 | Binding | Inhibition of MST1 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3745631 | single protein format | Scientific Literature | |
6. | ALA3748011 | Binding | Inhibition of human MST1 using [KKSRGDYMTMQIG] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
7. | ALA3760648 | Binding | Inhibition of MST1 (unknown origin) at 100 nM | Homo sapiens | 1 | ALA3758169 | single protein format | Scientific Literature | |
8. | ALA3777720 | Binding | Inhibition of N-terminal His6-tagged recombinant human MST1 expressed in baculovirus infected insect Sf9 cells assessed as remaining activity at 1 uM relative to control | Homo sapiens | 3 | ALA3774357 | cell-based format | Scientific Literature | |
9. | ALA3794938 | Binding | Inhibition of full length human N-terminal GST-tagged MST1 (1 to 487 residues) expressed in baculovirus expression system using fluorescence labelled IRS1 as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
10. | ALA3817274 | Binding | Inhibition of full length recombinant human GST-tagged MST1 expressed in baculovirus expression system at 1 uM relative to control | Homo sapiens | 1 | ALA3813614 | assay format | Scientific Literature | |
11. | ALA3817583 | Binding | Inhibition of human MST1 at 1 uM using [KKSRGDYMTMQIG] as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
12. | ALA3820255 | Binding | Inhibition of recombinant human full length GST-tagged MST1 expressed in Baculovirus at 1 uM relative to control | Homo sapiens | 1 | ALA3817726 | assay format | Scientific Literature | |
13. | ALA860661 | Binding | Average Binding Constant for STK4; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
14. | ALA1101778 | Binding | Inhibition of MST1 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
15. | ALA1116726 | Binding | Inhibition of MST1 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
16. | ALA1166578 | Binding | Inhibition of MST1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
17. | ALA1174925 | Binding | Inhibition of MST1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
18. | ALA1244302 | Binding | Inhibition of STK4 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
19. | ALA1244346 | Binding | Inhibition of STK4 | 1 | ALA1240341 | single protein format | Scientific Literature | ||
20. | ALA1244524 | Binding | Binding affinity to MST1 | 7 | ALA1240346 | single protein format | Scientific Literature |