# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA861048 | B | Average Binding Constant for PTK6; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
2. | ALA920661 | B | Inhibition of BRK | Homo sapiens | 1 | ALA1144565 | single protein format | Scientific Literature | |
3. | ALA928799 | B | Inhibition of Brk at 10 uM | 1 | ALA1141535 | single protein format | Scientific Literature | ||
4. | ALA927942 | B | Activity of human BRK kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
5. | ALA992508 | B | Inhibition of PTK6 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
6. | ALA988929 | B | Binding affinity to human BRK | Homo sapiens | 2 | ALA1151712 | single protein format | Scientific Literature | |
7. | ALA1035880 | B | Binding affinity to human BRK at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
8. | ALA953402 | B | Inhibition of Brk at 10 uM by HTRF assay relative to control | 57 | ALA1150387 | single protein format | Scientific Literature | ||
9. | ALA1060965 | B | Inhibition of BRK at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
10. | ALA1061159 | B | Binding constant for PTK6 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
11. | ALA1049963 | B | Binding affinity to BRK assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | ALA1154183 | single protein format | Scientific Literature | ||
12. | ALA1052938 | B | Inhibition of PTK6 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
13. | ALA1066616 | B | Residual activity of BRK at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
14. | ALA1047788 | B | Residual activity of BRK at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
15. | ALA1047815 | B | Residual activity of BRK at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
16. | ALA1066410 | B | Inhibition of recombinant BRK by TR-FRET assay | 3 | ALA1156877 | single protein format | Scientific Literature | ||
17. | ALA1072192 | B | Inhibition of BRK | 3 | ALA1157561 | single protein format | Scientific Literature | ||
18. | ALA1101497 | B | Inhibition of Brk at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
19. | ALA1107589 | B | Inhibition of BRK at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
20. | ALA1168803 | B | Inhibition of BRK at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature |