| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA861047 | B | Average Binding Constant for PKMYT1; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
| 2. | ALA920958 | B | Inhibition of Myt1 | 1 | ALA1145498 | single protein format | Scientific Literature | ||
| 3. | ALA981746 | B | Inhibition of PKMYT1 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
| 4. | ALA993457 | B | Binding affinity to human MYT1 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
| 5. | ALA1061154 | B | Binding constant for PKMYT1 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
| 6. | ALA1057598 | B | Inhibition of PKMYT1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
| 7. | ALA1166814 | B | Inhibition of PKMYT1 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
| 8. | ALA1175222 | B | Inhibition of PKMYT1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 9. | ALA1244372 | B | Inhibition of PKMYT1 | 1 | ALA1240341 | single protein format | Scientific Literature | ||
| 10. | ALA1244929 | B | Binding affinity to PKMYT1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 11. | ALA1798996 | B | Inhibition of MYT1 | 1 | ALA1795201 | single protein format | Scientific Literature | ||
| 12. | ALA1826613 | B | Activity of PKMYT1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 13. | ALA1908454 | B | Binding constant for PKMYT1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 14. | ALA1948657 | B | Activity at full length human Myt1 expressed in human HEK293 cells at 10 uM after 30 mins by fluorescence polarization immunoassay | Homo sapiens | 1 | ALA1944550 | cell-based format | Scientific Literature | |
| 15. | ALA1948658 | B | Competitive inhibition of human Myt1 by TR-FRET assay | Homo sapiens | 2 | ALA1944550 | single protein format | Scientific Literature | |
| 16. | ALA1948659 | B | Activity at full length human Myt1 expressed in human HEK293 cells assessed as Cdk1 phosphorylation at Try15 at 10 uM after 30 mins by fluorescence polarization immunoassay | Homo sapiens | 5 | ALA1944550 | cell-based format | Scientific Literature | |
| 17. | ALA1948660 | B | Activity at full length human Myt1 expressed in human HEK293 cells assessed as Cdk1 phosphorylation at Thr14 at 10 uM after 30 mins by fluorescence polarization immunoassay | Homo sapiens | 5 | ALA1944550 | cell-based format | Scientific Literature | |
| 18. | ALA1948661 | B | Activity at human Myt1 (75 to 362) expressed in Escherichia coli BL21 (DE3) cells assessed as Cdk1 phosphorylation at Try15 at 10 uM after 30 mins by fluorescence polarization immunoassay | Homo sapiens | 5 | ALA1944550 | cell-based format | Scientific Literature | |
| 19. | ALA1948662 | B | Activity at human Myt1 (75 to 362) expressed in Escherichia coli BL21 (DE3) cells assessed as Cdk1 phosphorylation at Thr14 at 10 uM after 30 mins by fluorescence polarization immunoassay | Homo sapiens | 5 | ALA1944550 | cell-based format | Scientific Literature | |
| 20. | ALA1959385 | B | Inhibition of PKMYT1 at 1 uM | 1 | ALA1955770 | single protein format | Scientific Literature |
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