# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3578904 | Binding | Competitive binding affinity to KHS1 in human A375 cells after 15 mins in presence of ATP analogue | Homo sapiens | 1 | ALA3576847 | cell-based format | Scientific Literature | |
2. | ALA3595429 | Binding | Inhibition of recombinant human KHS1 at 1 uM relative to control | Homo sapiens | 1 | ALA3593241 | single protein format | Scientific Literature | |
3. | ALA3631269 | Binding | Inhibition of KHS (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
4. | ALA3742712 | Binding | Inhibition of KHS (unknown origin) | Homo sapiens | 1 | ALA3739276 | single protein format | Scientific Literature | |
5. | ALA3751067 | Binding | Inhibition of KHS1 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3745631 | single protein format | Scientific Literature | |
6. | ALA3748231 | Binding | Inhibition of human KHS using MBP as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
7. | ALA3762903 | Binding | Inhibition of KHS1 (unknown origin) at 100 nM | Homo sapiens | 1 | ALA3758169 | single protein format | Scientific Literature | |
8. | ALA3772530 | Binding | Inhibition of human recombinant KHS1 | Homo sapiens | 1 | ALA3769359 | single protein format | Scientific Literature | |
9. | ALA3772905 | Binding | Inhibition of human recombinant KHS1 at 0.1 uM | Homo sapiens | 1 | ALA3769359 | single protein format | Scientific Literature | |
10. | ALA3816716 | Binding | Inhibition of human KHS at 1 uM using MBP as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
11. | ALA3817254 | Binding | Inhibition of full length recombinant human GST-tagged KHS1 expressed in baculovirus expression system at 1 uM relative to control | Homo sapiens | 1 | ALA3813614 | assay format | Scientific Literature | |
12. | ALA3820369 | Binding | Inhibition of recombinant human full length GST-tagged KHS1 expressed in Baculovirus at 1 uM relative to control | Homo sapiens | 2 | ALA3817726 | assay format | Scientific Literature | |
13. | ALA860642 | Binding | Average Binding Constant for MAP4K5; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
14. | ALA1166063 | Binding | Inhibition of MAP4K5 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
15. | ALA1174896 | Binding | Inhibition of MAP4K5 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
16. | ALA1219793 | Binding | Inhibition of MAP4K5 at 1 uM by radiometric method | 2 | ALA1212904 | single protein format | Scientific Literature | ||
17. | ALA1244206 | Binding | Inhibition of MAP4K5 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
18. | ALA1244320 | Binding | Inhibition of MAP4K5 | 1 | ALA1240341 | single protein format | Scientific Literature | ||
19. | ALA1244497 | Binding | Binding affinity to MAP4K5 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
20. | ALA1252477 | Binding | Inhibition of MAP4K5 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature |