| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA714431 | F | Antagonist activity against muscarinic M1 receptor from rabbit vas deferens | Oryctolagus cuniculus | 40 | ALA1126608 | tissue-based format | Scientific Literature | |
| 2. | ALA747252 | F | Potency at ganglionic muscarinic acetylcholine receptor M1 mediating tachycardia to increase the heart rate in pithed rat | Cavia porcellus | 1 | ALA1125528 | tissue-based format | Scientific Literature | |
| 3. | ALA747253 | B | Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M1 | Cavia porcellus | 4 | ALA1128457 | single protein format | Scientific Literature | |
| 4. | ALA747254 | B | The compound was tested for Antimuscarinic activity against muscarinic acetylcholine receptor M1 from vas deferens of rabbit | Cavia porcellus | 1 | ALA1126261 | single protein format | Scientific Literature | |
| 5. | ALA747393 | B | Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]QNB from guinea pig cerebral cortex | Cavia porcellus | 37 | ALA1128229 | tissue-based format | Scientific Literature | |
| 6. | ALA747394 | B | Compound was evaluated for its binding affinity against Muscarinic acetylcholine receptor M1 in guinea pig cerebral cortex using (-)-[3H]-QNB as radioligand | Cavia porcellus | 2 | ALA1126289 | tissue-based format | Scientific Literature | |
| 7. | ALA747395 | B | Compound was evaluated for its binding affinity against muscarinic acetylcholine receptor M1 in guinea pig cerebral cortex using (-)-[3H]-QNB as radioligand | Cavia porcellus | 6 | ALA1126289 | tissue-based format | Scientific Literature | |
| 8. | ALA857139 | F | Antagonistic potency against Muscarinic acetylcholine receptor M1 (10 uM) | Cavia porcellus | 2 | ALA1131149 | assay format | Scientific Literature | |
| 9. | ALA747396 | F | Antagonistic potency against Muscarinic acetylcholine receptor M1; nd= Not determined | Cavia porcellus | 9 | ALA1131149 | assay format | Scientific Literature | |
| 10. | ALA747397 | B | Inhibition of [3H]QNB binding to CHO cells bearing transfected muscarinic acetylcholine receptor M1 | Cricetulus griseus | 1 | ALA1125674 | cell-based format | Scientific Literature | |
| 11. | ALA747398 | B | Inhibition of [3H]QNB binding to CHO cells bearing transfected muscarinic acetylcholine receptor M3 | Cricetulus griseus | 1 | ALA1125674 | cell-based format | Scientific Literature | |
| 12. | ALA750971 | B | Ability to stimulate biochemical responses in cell lines expressing muscarinic A9 L receptor sub types | 9 | ALA1145111 | cell-based format | Scientific Literature | ||
| 13. | ALA750972 | B | Ability to stimulate biochemical responses in cell lines expressing muscarinic A9 L receptor sub types; Not determined | 2 | ALA1145111 | cell-based format | Scientific Literature | ||
| 14. | ALA750973 | B | Binding affinity at the NMS liganded human muscarinic acetylcholine receptor M1 was estimated as log affinity (log1/M) | 24 | ALA1132569 | single protein format | Scientific Literature | ||
| 15. | ALA750974 | B | Binding affinity at the unliganded human muscarinic acetylcholine receptor M1 was estimated as log affinity (log1/M) | 24 | ALA1132569 | single protein format | Scientific Literature | ||
| 16. | ALA882645 | F | Evaluated for its HMPA (human muscarinic inositol phosphate accumulation) activity measured in CHO cells expressing Muscarinic acetylcholine receptor M1 compound run at 100 uM | 11 | ALA1150001 | cell-based format | Scientific Literature | ||
| 17. | ALA750975 | F | Evaluated for its HMPA (human muscarinic inositol phosphate accumulation) activity measured in CHO cells expressing Muscarinic acetylcholine receptor M1 compound run at 100 uM; 100 uM of carbachol was used; No data | 1 | ALA1150001 | cell-based format | Scientific Literature | ||
| 18. | ALA750976 | F | Maximal response obtained for each drug normalized to effect of carbachol in Muscarinic acetylcholine receptor M1 | 3 | ALA1131286 | assay format | Scientific Literature | ||
| 19. | ALA752214 | F | Stimulation of inositol phosphate(PI) accumulation in CHO cells expressing Muscarinic acetylcholine receptor M1 as maximal response at 100 uM relative to carbachol | Homo sapiens | 10 | ALA1131286 | cell-based format | Scientific Literature | |
| 20. | ALA752215 | F | Stimulations of inositol phosphate(PI) accumulation in transfected CHO cells in Muscarinic acetylcholine receptor M1 values are the maximal response obtained from the compound tested at 100 uM normalized to the effects of carbachol. | 1 | ALA1131286 | cell-based format | Scientific Literature |
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