# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA677252 | B | In vitro inhibition of non-cytotoxic immunophilin FK506 binding protein activity | Homo sapiens | 17 | single protein format | Scientific Literature | ||
2. | ALA682210 | B | Inhibition of peptidyl-prolyl isomerase (PPIase, or rotamase) activity of FK506 binding protein 12 | 40 | single protein format | Scientific Literature | |||
3. | ALA682211 | B | Ability to inhibit peptidyl-prolyl isomerase (PPIase, or rotamase) activity of FK506 binding protein 12 | 53 | single protein format | Scientific Literature | |||
4. | ALA682212 | B | Effective concentration determined was towards FK506 binding protein 12 by competitive binding assay using [3H]-dihydro FK-506 as radioligand | 5 | single protein format | Scientific Literature | |||
5. | ALA678139 | B | Effective concentration against FK506 binding protein 12 using [3H]-dihydro FK-506 | Homo sapiens | 11 | single protein format | Scientific Literature | ||
6. | ALA678140 | B | Compound was evaluated for its inhibitory effect on human FK506 binding protein 12 by means of protease-coupled PPIase assay | 10 | single protein format | Scientific Literature | |||
7. | ALA678141 | B | Inhibitory binding activity against human Immunophilin-FK-506 binding protein 12 | 27 | single protein format | Scientific Literature | |||
8. | ALA678142 | B | The compound was tested for binding affinity against human FK506 binding protein 12 | 4 | single protein format | Scientific Literature | |||
9. | ALA678143 | B | Compound was tested for its ability to inhibit FK506 binding protein 12 rotamase activity | 67 | single protein format | Scientific Literature | |||
10. | ALA678144 | B | Inhibition constant(Ki) for inhibition of PPIase activity of human FK506 binding protein 12 (Conc=14 nM) of FKBPs family | 1 | single protein format | Scientific Literature | |||
11. | ALA678145 | B | Inhibitory activity against FK506 binding protein 12 | Homo sapiens | 11 | single protein format | Scientific Literature | ||
12. | ALA857528 | B | Apparent inhibition constant of Wild-type human recombinant FK506 binding protein 12 | 17 | single protein format | Scientific Literature | |||
13. | ALA678146 | B | Inhibitory activity of compound against FK506 binding protein 12 was determined | 6 | single protein format | Scientific Literature | |||
14. | ALA678147 | F | Inhibitory selectivity for human FK506 binding protein 12 and human mixed lymphocyte response(MLR) | Homo sapiens | 27 | assay format | Scientific Literature | ||
15. | ALA678148 | B | Immunosuppressive activity in FK506 binding protein 12 binding assay as inhibitory concentration (rIC50) relative to FK506 IC50 (1.2 nM) | Homo sapiens | 11 | single protein format | Scientific Literature | ||
16. | ALA678150 | B | Ability to bind the major cystolic receptor FK506 binding protein 12 by using competitive binding assay | 4 | single protein format | Scientific Literature | |||
17. | ALA678151 | B | Ability to bind the major cystolic receptor FK506 binding protein 12 by using competitive binding assay | 16 | single protein format | Scientific Literature | |||
18. | ALA678152 | B | Ability to bind the major cystolic receptor FK506 binding protein 12 by using competitive binding assay; No data | 1 | single protein format | Scientific Literature | |||
19. | ALA678153 | B | Ability to bind the major cystolic receptor FKBP12 by using competitive binding assay | 1 | single protein format | Scientific Literature | |||
20. | ALA678154 | B | Binding affinity for FK506 binding protein 12 using [3H]-dihydro FK-506 radioligand was determined | 5 | single protein format | Scientific Literature |