DCLK1-IN-1 , CAS No.D609779, Inhibitor of doublecortin like kinase 1;Inhibitor of doublecortin like kinase 2;Inhibitor of leucine rich repeat kinase 2;Inhibitor of mitogen-activated protein kinase 7
DCLK1-IN-1 , CAS No.D609779, Inhibitor of doublecortin like kinase 1;Inhibitor of doublecortin like kinase 2;Inhibitor of leucine rich repeat kinase 2;Inhibitor of mitogen-activated protein kinase 7
Inhibitor of doublecortin like kinase 1;Inhibitor of doublecortin like kinase 2;Inhibitor of leucine rich repeat kinase 2;Inhibitor of mitogen-activated protein kinase 7
1.Ferguson FM, Nabet B, Raghavan S, Liu Y, Leggett AL, Kuljanin M, Kalekar RL, Yang A, He S, Wang J et al.. (2020) Discovery of a selective inhibitor of doublecortin like kinase 1.. Nat Chem Biol, 16 (6):(635-643). [PMID:32251410]
2.Ferguson FM, Liu Y, Harshbarger W, Huang L, Wang J, Deng X, Capuzzi SJ, Muratov EN, Tropsha A, Muthuswamy S et al.. (2020) Synthesis and Structure-Activity Relationships of DCLK1 Kinase Inhibitors Based on a 5,11-Dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-one Scaffold.. J Med Chem, 63 (14):(7817-7826). [PMID:32530623]
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