enclomiphene , Estrogen receptor alpha modulator, CAS No.15690-57-0, Estrogen receptor alpha modulator

Item Number

E610124

Grouped product items
SKU	Size	Availability	Price
E610124-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$46.90
E610124-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$69.90
E610124-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$129.90
E610124-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$219.90
E610124-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$329.90
E610124-250mg	250mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$579.90
E610124-1g	1g	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,623.90

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Basic Description

Synonyms	Enclomiphene\|clomiphene\|Clomifene\|trans-Clomiphene\|Enclomifene\|15690-57-0\|trans-Clomifene\|Enclomiphene [USAN]\|ISOMER B\|RMI 16,289\|Cisclomiphene\|Enclomifene [INN]\|Clomiphene trans-form\|ISOMER-B\|R6D2UI4FLS\|Clomifeno\|(E)-2-(p-(2-Chloro-1,2-diphenylvinyl)phen
Specifications & Purity	Moligand™, ≥98%
Storage Temp	Store at 2-8°C,Protected from light
Shipped In	Wet ice
Grade	Moligand™
Action Type	MODULATOR
Mechanism of action	Estrogen receptor alpha modulator
Product Description	Enclomiphene ((E)-Clomiphene) is a potent and orally active non-steroidal estrogen receptor antagonist, with antioestrogenic property. Enclomiphene can be used for the research of ovarian dysfunction, testosterone deficiency, male hypogonadism and type 2 diabetes.

Names and Identifiers

IUPAC Name	2-[4-[(E)-2-chloro-1,2-diphenylethenyl]phenoxy]-N,N-diethylethanamine
INCHI	InChI=1S/C26H28ClNO/c1-3-28(4-2)19-20-29-24-17-15-22(16-18-24)25(21-11-7-5-8-12-21)26(27)23-13-9-6-10-14-23/h5-18H,3-4,19-20H2,1-2H3/b26-25+
InChi Key	GKIRPKYJQBWNGO-OCEACIFDSA-N
Canonical SMILES	CCN(CC)CCOC1=CC=C(C=C1)C(=C(C2=CC=CC=C2)Cl)C3=CC=CC=C3
Isomeric SMILES	CCN(CC)CCOC1=CC=C(C=C1)/C(=C(\C2=CC=CC=C2)/Cl)/C3=CC=CC=C3
PubChem CID	1548953
Molecular Weight	405.96

PubChem CID

ChEMBL Ligand

CAS Registry No.

RCSB PDB Ligand

References

1. Ioannidou-Kadis S, Wright PJ, Neely RD, Quinton R. (2006) Complete reversal of adult-onset isolated hypogonadotropic hypogonadism with clomiphene citrate.. Fertil Steril, 86 (5): (1513.e5-9). [PMID:17070201]
2. Hill S, Arutchelvam V, Quinton R. (2009) Enclomiphene, an estrogen receptor antagonist for the treatment of testosterone deficiency in men.. IDrugs, 12 (2): (109-19). [PMID:19204885]

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Basic Description