Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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F335497-5mg | 5mg | In stock | $213.90 | |
F335497-10mg | 10mg | In stock | $384.90 | |
F335497-25mg | 25mg | In stock | $865.90 | |
F335497-50mg | 50mg | In stock | $1,558.90 | |
F335497-100mg | 100mg | In stock | $2,804.90 |
a highly selective D4 dopamine receptor full antagonist
Synonyms | FAUC 213|337972-47-1|FAUC-213|FAUC213|2-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine|CHEMBL310843|G8F040299R|2-((4-(4-Chlorophenyl)piperazin-1-yl)methyl)pyrazolo[1,5-a]pyridine|2-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]pyrazolo[1,5-a] |
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Specifications & Purity | Moligand™, ≥98% |
Storage Temp | Store at 2-8°C |
Shipped In | Wet ice |
Grade | Moligand™ |
Action Type | AGONIST, ANTAGONIST |
Mechanism of action | Agonist of D 4 receptor;Antagonist of D 4 receptor |
Product Description | FAUC 213 is a highly selective D4 dopamine receptor full antagonist. |
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IUPAC Name | 2-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]pyrazolo[1,5-a]pyridine |
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INCHI | InChI=1S/C18H19ClN4/c19-15-4-6-17(7-5-15)22-11-9-21(10-12-22)14-16-13-18-3-1-2-8-23(18)20-16/h1-8,13H,9-12,14H2 |
InChi Key | DTRXURJDKOYCCD-UHFFFAOYSA-N |
Canonical SMILES | C1CN(CCN1CC2=NN3C=CC=CC3=C2)C4=CC=C(C=C4)Cl |
Isomeric SMILES | C1CN(CCN1CC2=NN3C=CC=CC3=C2)C4=CC=C(C=C4)Cl |
PubChem CID | 10336538 |
Molecular Weight | 326.82 |
PubChem CID | 10336538 |
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ChEMBL Ligand | CHEMBL310843 |
BindingDB Ligand | 50102712 |
CAS Registry No. | 337972-47-1 |
GPCRdb Ligand | FAUC213 |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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I2222599 | Certificate of Analysis | Jul 20, 2022 | F335497 |
I2222600 | Certificate of Analysis | Jul 20, 2022 | F335497 |
I2222612 | Certificate of Analysis | Jul 20, 2022 | F335497 |
I2222614 | Certificate of Analysis | Jul 20, 2022 | F335497 |
I2222615 | Certificate of Analysis | Jul 20, 2022 | F335497 |
Solubility | Soluble in DMSO: ~24 mg/mL with warming up to 60° C: water: insoluble |
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Pictogram(s) | GHS07 |
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Signal | Warning |
Hazard Statements | H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation |
Precautionary Statements | P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing. P280:Wear protective gloves/protective clothing/eye protection/face protection. P302+P352:IF ON SKIN: wash with plenty of water. P321:Specific treatment (see ... on this label). P405:Store locked up. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P271:Use only outdoors or in a well-ventilated area. P304+P340:IF INHALED: Remove person to fresh air and keep comfortable for breathing. P403+P233:Store in a well-ventilated place. Keep container tightly closed. P362+P364:Take off contaminated clothing and wash it before reuse. P264+P265:Wash hands [and …] thoroughly after handling. Do not touch eyes. P337+P317:If eye irritation persists: Get medical help. P332+P317:If skin irritation occurs: Get medical help. P319:Get medical help if you feel unwell. |