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GNTI dihydrochloride - ≥96%(HPLC), high purity , CAS No.351183-88-5

Item Number

G287224

Grouped product items
SKU	Size	Availability	Price	Qty
G287224-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$199.90
G287224-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$838.90

Potent, selective κ antagonist

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Basic Description

Specifications & Purity	≥96%(HPLC)
Biochemical and Physiological Mechanisms	Highly potentκopioid receptor antagonist (Ki= 0.18 nM for human clonedκreceptors expressed in CHO cells). Displays 208- and 799-fold selectivity overμandδreceptors respectively. Reduces feeding behavior in rats with a much higher potency (300-30,000-fold)
Storage Temp	Store at -20°C,Desiccated
Shipped In	Ice chest + Ice pads

InChi Key	GJPIMNXJPMPQHK-CVVXFVLRSA-N
Canonical SMILES	OC3=CC=C2CC([C@@]5(O)[C@@]4(CC8)C2=C3O[C@H]4C(NC7=C6C=C(NC=N)C=C7)=C6C5)N8CC1CC1.Cl.Cl
Isomeric SMILES	C1CC1CN2CC[C@]34[C@@H]5C6=C(C[C@]3(C2CC7=C4C(=C(C=C7)O)O5)O)C8=C(N6)C=CC(=C8)N=CN.Cl.Cl
PubChem CID	90479777
Molecular Weight	544.48

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Solubility	Solvent:water, Max Conc. mg/mL: 54.45, Max Conc. mM: 100; Solvent:DMSO, Max Conc. mg/mL: 54.45, Max Conc. mM: 100

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