Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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G129271-5mg | 5mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $28.90 | |
G129271-25mg | 25mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $117.90 | |
G129271-100mg | 100mg | In stock | $391.90 | |
G129271-250mg | 250mg | In stock | $882.90 | |
G129271-1g | 1g | In stock | $3,175.90 | |
G129271-5g | 5g | In stock | $14,288.90 |
General serine protease inhibitor
Synonyms | Gabexate mesylate|56974-61-9|Gabexate mesilate|Gabexate (mesylate)|Gabexate Methanesulfonate|FOY|56974-61-9 (mesylate)|Gabexate mesilate [JAN]|CHEMBL1398351|DTXSID0045591|NCGC00017121-01|ethyl 4-((6-guanidinohexanoyl)oxy)benzoate methanesulfonate|CAS-5697 |
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Specifications & Purity | ≥99% |
Biochemical and Physiological Mechanisms | General serine protease inhibitor (K i values are 3.4 nM, 5, 1.8 µM and 2.6 mM at tryptase, thrombin, tyrpsin and kallikrein serine proteases respectively). Additionally inhibits nitric oxide synthase. Displays antithrombotic activity and antitumor effect |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Note | 5mg卖完停产,不再备货。Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details. |
Product Description | Gabexate mesylate |
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IUPAC Name | ethyl 4-[6-(diaminomethylideneamino)hexanoyloxy]benzoate;methanesulfonic acid |
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INCHI | InChI=1S/C16H23N3O4.CH4O3S/c1-2-22-15(21)12-7-9-13(10-8-12)23-14(20)6-4-3-5-11-19-16(17)18;1-5(2,3)4/h7-10H,2-6,11H2,1H3,(H4,17,18,19);1H3,(H,2,3,4) |
InChi Key | DNTNDFLIKUKKOC-UHFFFAOYSA-N |
Canonical SMILES | CCOC(=O)C1=CC=C(C=C1)OC(=O)CCCCCN=C(N)N.CS(=O)(=O)O |
Isomeric SMILES | CCOC(=O)C1=CC=C(C=C1)OC(=O)CCCCCN=C(N)N.CS(=O)(=O)O |
PubChem CID | 6604561 |
Molecular Weight | 417.48 |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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I2227298 | Certificate of Analysis | Jul 15, 2024 | G129271 |
I2227299 | Certificate of Analysis | Jul 15, 2024 | G129271 |
I2227300 | Certificate of Analysis | Jul 15, 2024 | G129271 |
I2227303 | Certificate of Analysis | Jul 15, 2024 | G129271 |
H1520105 | Certificate of Analysis | Mar 09, 2023 | G129271 |
D2222114 | Certificate of Analysis | May 02, 2022 | G129271 |
D2222123 | Certificate of Analysis | May 02, 2022 | G129271 |
D2222125 | Certificate of Analysis | May 02, 2022 | G129271 |
Solubility | DMSO 83 mg/mL Water 12 mg/mL Ethanol 83 mg/mL |
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Melt Point(°C) | 91 °C |
Merck Index | 4320 |
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