Click Here for 5% Off Your First Aladdin Purchase!

Gisadenafil - ≥98%, high purity , Phosphodiesterase 5A inhibitor, CAS No.334826-98-1, Phosphodiesterase 5A inhibitor

  • Moligand™
  • ≥98%
Item Number
G610562
Grouped product items
SKUSizeAvailabilityPrice Qty
G610562-1mg
1mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$189.90
G610562-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$304.90
G610562-10mg
10mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$639.90
G610562-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,060.90
G610562-50mg
50mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,299.90
View related series
phosphodiesterase 5A Inhibitor

Basic Description

SynonymsGISADENAFIL|334826-98-1|UNII-S6G4R7DI1C|Gisadenafil [USAN:INN]|S6G4R7DI1C|UK-369,003|5-[2-Ethoxy-5-(4-ethylpiperazin-1-ylsulfonyl)pyridin-3-yl]-3-ethyl-2-(2-methoxyethyl)-2,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-one|UK 369003|UK-369003|CHEMBL1928262|UK03
Specifications & PurityMoligand™, ≥98%
Biochemical and Physiological MechanismsGisadenafil (UK-369003) is a specific, orally active phosphodiesterase 5 (PDE5) inhibitor with an IC50 of 3.6 nM and prevents degradation of cyclic guanosine monophosphate (cGMP).
Storage TempStore at -20°C
Shipped InIce chest + Ice pads
GradeMoligand™
Action TypeINHIBITOR
Mechanism of actionPhosphodiesterase 5A inhibitor

Product Properties

ALogP0.5

Associated Targets

PDE5A Tclin cGMP-specific 3',5'-cyclic phosphodiesterase 2 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

IUPAC Name 5-[2-ethoxy-5-(4-ethylpiperazin-1-yl)sulfonylpyridin-3-yl]-3-ethyl-2-(2-methoxyethyl)-4H-pyrazolo[3,4-e]pyrimidin-7-one
INCHI InChI=1S/C23H33N7O5S/c1-5-18-19-20(27-30(18)12-13-34-4)22(31)26-21(25-19)17-14-16(15-24-23(17)35-7-3)36(32,33)29-10-8-28(6-2)9-11-29/h14-15H,5-13H2,1-4H3,(H,25,26,31)
InChi Key YPFZMBHKIVDSNR-UHFFFAOYSA-N
Canonical SMILES COCCn1nc2c(c1CC)[nH]c(nc2=O)c1cc(cnc1OCC)S(=O)(=O)N1CCN(CC1)CC
Isomeric SMILES CCC1=C2C(=NN1CCOC)C(=O)NC(=N2)C3=C(N=CC(=C3)S(=O)(=O)N4CCN(CC4)CC)OCC
PubChem CID 135536943
Molecular Weight 519.62

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

Related Documents

Solution Calculators