GLPG3970 , CAS No.2403733-82-2, Inhibitor of salt inducible kinase 2;Inhibitor of SIK family kinase 3

Item Number

G610582

Grouped product items
SKU	Size	Availability	Price	Qty
G610582-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$350.90
G610582-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,200.90

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Basic Description

Synonyms	GLPG3970\|GLPG-3970\|UA6B2TI4MO\|UNII-UA6B2TI4MO\|2403733-82-2\|1(2H)-Isoquinolinone, 3,4-dihydro-8-methoxy-6-(7-(2-(4-morpholinyl)ethoxy)imidazo(1,2-a)pyridin-3-yl)-2-(2,2,2-trifluoroethyl)-\|8-Methoxy-6-[7-(2-morpholin-4-ylethoxy)imidazo[1,2-a]pyridin-3-yl]-2
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of salt inducible kinase 2;Inhibitor of SIK family kinase 3

Associated Targets

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	8-methoxy-6-[7-(2-morpholin-4-ylethoxy)imidazo[1,2-a]pyridin-3-yl]-2-(2,2,2-trifluoroethyl)-3,4-dihydroisoquinolin-1-one
INCHI	InChI=1S/C25H27F3N4O4/c1-34-21-13-18(12-17-2-4-31(16-25(26,27)28)24(33)23(17)21)20-15-29-22-14-19(3-5-32(20)22)36-11-8-30-6-9-35-10-7-30/h3,5,12-15H,2,4,6-11,16H2,1H3
InChi Key	XASOHFCUIQARJT-UHFFFAOYSA-N
Canonical SMILES	COc1cc(cc2c1C(=O)N(CC2)CC(F)(F)F)c1cnc2n1ccc(c2)OCCN1CCOCC1
Isomeric SMILES	COC1=CC(=CC2=C1C(=O)N(CC2)CC(F)(F)F)C3=CN=C4N3C=CC(=C4)OCCN5CCOCC5
PubChem CID	146273261

PubChem CID

CAS Registry No.

ChEMBL Ligand

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Basic Description