| SKU | Size | Availability | Price | Qty |
|---|---|---|---|---|
| G655301-1ml | 1ml | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $77.90 |
| Specifications & Purity | 10mM in DMSO |
|---|---|
| Storage Temp | Store at -80°C |
| Shipped In | Ice chest + Ice pads |
| Product Description | GPR52 antagonist-1 (Compound 43) is a GPR52 antagonist with an IC 50 of 0.63 μM. GPR52 antagonist-1 reduces mHTT (mutant huntingtin protein) levels by targeting GPR52 and promotes survival of mouse primary striatal neurons In Vivo GPR52 antagonist-1 (Compound 43) (5 mg/kg; i.p.; once a day for 4 weeks) reduces mHTT levels and rescues HD-related phenotypes in HdhQ140 mice . MCE has not independently confirmed the accuracy of these methods. They are for reference only. IC50& Target:IC 50 : 0.63 μM (GPR52) |
| Canonical SMILES | C1=CC=C(C=C1)CCC=CC(=O)C2=CC=CS2 |
|---|---|
| Molecular Weight | 242.34 |
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