Granisetron - ≥98.0%, high purity , CAS No.109889-09-0, Antagonist of 5-HT 3A

Item Number

G127257

Grouped product items
SKU	Size	Availability	Price
G127257-5mg	5mg	In stock	$68.90
G127257-25mg	25mg	In stock	$240.90
G127257-100mg	100mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$686.90
G127257-250mg	250mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$1,201.90

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Basic Description

Synonyms	granisetron\|109889-09-0\|Sancuso\|Sustol\|Kevatril\|Granisetronum\|APF530\|Kytril\|BRL-43694\|1-methyl-N-[(1S,5R)-9-methyl-9-azabicyclo[3.3.1]nonan-3-yl]indazole-3-carboxamide\|CHEBI:5537\|BRL 43694\|APF 530\|WZG3J2MCOL\|1-methyl-N-[(3-endo)-9-methyl-9-azabicyclo[3.3.
Specifications & Purity	≥98.0%
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of 5-HT 3A
Product Description	Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy.

Names and Identifiers

IUPAC Name	1-methyl-N-[(1R,5S)-9-methyl-9-azabicyclo[3.3.1]nonan-3-yl]indazole-3-carboxamide
INCHI	InChI=1S/C18H24N4O/c1-21-13-6-5-7-14(21)11-12(10-13)19-18(23)17-15-8-3-4-9-16(15)22(2)20-17/h3-4,8-9,12-14H,5-7,10-11H2,1-2H3,(H,19,23)/t12?,13-,14+
InChi Key	MFWNKCLOYSRHCJ-AGUYFDCRSA-N
Canonical SMILES	CN1C2CCCC1CC(C2)NC(=O)C3=NN(C4=CC=CC=C43)C
Isomeric SMILES	CN1[C@@H]2CCC[C@H]1CC(C2)NC(=O)C3=NN(C4=CC=CC=C43)C
PubChem CID	5284566
Molecular Weight	312.41

DrugBank Ligand

Wikipedia

CAS Registry No.

PubChem CID

Certificates

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4 results found

Lot Number	Certificate Type	Date	Item
J2022133	Certificate of Analysis	Aug 12, 2022	G127257
J2022132	Certificate of Analysis	Aug 12, 2022	G127257
J2022131	Certificate of Analysis	Aug 12, 2022	G127257
J2022130	Certificate of Analysis	Aug 12, 2022	G127257

Safety and Hazards(GHS)

Pictogram(s)	GHS07
Signal	Warning
Hazard Statements	H319:Causes serious eye irritation H412:Harmful to aquatic life with long lasting effects H302:Harmful if swallowed
Precautionary Statements	P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing. P273:Avoid release to the environment. P280:Wear protective gloves/protective clothing/eye protection/face protection. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P330:Rinse mouth. P264+P265:Wash hands [and …] thoroughly after handling. Do not touch eyes. P301+P317:IF SWALLOWED: Get medical help. P337+P317:If eye irritation persists: Get medical help.

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Basic Description