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GSK-Bz derivative 2b , CAS No.G610738, Inhibitor of TRPV4

Item Number

G610738

Grouped product items
SKU	Size	Availability	Price	Qty
G610738-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$572.90
G610738-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	N-(5,6-dichloro-1-{1-[4-(1-cyanocyclobutyl)phenyl]piperidin-4-yl}-2-[(propan-2-yl)amino]-1H-1,3-benzodiazol-4-yl)acetamide
INCHI	InChI=1S/C28H32Cl2N6O/c1-17(2)32-27-34-25-23(15-22(29)24(30)26(25)33-18(3)37)36(27)21-9-13-35(14-10-21)20-7-5-19(6-8-20)28(16-31)11-4-12-28/h5-8,15,17,21H,4,9-14H2,1-3H3,(H,32,34)(H,33,37)
InChi Key	HKOYZUBWZOWYKY-UHFFFAOYSA-N
Canonical SMILES	CC(C)NC1=NC2=C(C=C(Cl)C(Cl)=C2NC(C)=O)N1C3CCN(CC3)C4=CC=C(C=C4)C5(CCC5)C#N

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1. Ai C, Wang Z, Li P, Wang M, Zhang W, Song H, Cai X, Lv K, Chen X, Zheng Z. (2023) Discovery and pharmacological characterization of a novel benzimidazole TRPV4 antagonist with cyanocyclobutyl moiety.. Eur J Med Chem, 249 (3): (115137). [PMID:36696767]

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