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GSK2798745 , CAS No.G610709, Inhibitor of TRPV4

Item Number

G610709

Grouped product items
SKU	Size	Availability	Price	Qty
G610709-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
G610709-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,334.90

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Basic Description

Synonyms	GSK2798745\|1419609-94-1\|UNII-63FJ7LF55O\|GSK-2798745\|63FJ7LF55O\|3-[[(5S,7S)-3-[5-(2-hydroxypropan-2-yl)pyrazin-2-yl]-7-methyl-2-oxo-1-oxa-3-azaspiro[4.5]decan-7-yl]methyl]benzimidazole-5-carbonitrile\|CHEMBL4470585\|1-(((5S,7S)-3-(5-(2-Hydroxypropan-2-yl)pyr
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of TRPV4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	3-[[(5S,7S)-3-[5-(2-hydroxypropan-2-yl)pyrazin-2-yl]-7-methyl-2-oxo-1-oxa-3-azaspiro[4.5]decan-7-yl]methyl]benzimidazole-5-carbonitrile
INCHI	InChI=1S/C25H28N6O3/c1-23(2,33)20-11-28-21(12-27-20)31-15-25(34-22(31)32)8-4-7-24(3,13-25)14-30-16-29-18-6-5-17(10-26)9-19(18)30/h5-6,9,11-12,16,33H,4,7-8,13-15H2,1-3H3/t24-,25-/m0/s1
InChi Key	URCMKDJBULWNAI-DQEYMECFSA-N
Canonical SMILES	C[C@@]1(CCC[C@]2(C1)CN(C(=O)O2)C3=NC=C(N=C3)C(C)(C)O)CN4C=NC5=C4C=C(C=C5)C#N
Isomeric SMILES	C[C@@]1(CCC[C@]2(C1)CN(C(=O)O2)C3=NC=C(N=C3)C(C)(C)O)CN4C=NC5=C4C=C(C=C5)C#N
PubChem CID	71227359

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