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[³H]dizocilpine , CAS No.H614101, Antagonist of GluN1;Channel blocker of GluN2A;Channel blocker of GluN2B;Channel blocker of GluN2C;Channel blocker of GluN2D

Moligand™

PubChem CID: 1207

Item Number

H614101

Grouped product items
SKU	Size	Availability	Price	Qty
H614101-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
H614101-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,001.90

View related series

GluN1 Antagonist GluN2A Channel blocker GluN2B Channel blocker GluN2C Channel blocker GluN2D Channel blocker

Basic Description

Synonyms	70449-94-4\|Neurogard\|(+)-MK 801\|10,11-dihydro-5-methyl-5h-dibenzo[a,d]cyclohepten-5,10-imine\|[3H]MK-801\|MK-801\|5-methyl-10,11-dihydro-5H-5,10-epiminodibenzo[a,d][7]annulene\|MK801\|10,11-Dihydro-5-methyl-5H-dibenzo(a,d)cyclohepten-5,10-imine\|[3H]dizocilpine
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	ANTAGONIST, CHANNEL BLOCKER
Mechanism of action	Antagonist of GluN1;Channel blocker of GluN2A;Channel blocker of GluN2B;Channel blocker of GluN2C;Channel blocker of GluN2D

Associated Targets

TXNRD1 Tclin Thioredoxin reductase 1, cytoplasmic 0 Activities

Discover Target: TXNRD1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

RGS4 Tchem Regulator of G-protein signaling 4 0 Activities

Discover Target: RGS4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

ATXN2 Tbio Ataxin-2 0 Activities

Discover Target: ATXN2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIN1 Tclin Glutamate receptor ionotropic, NMDA 1 0 Activities

Discover Target: GRIN1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIN2A Tclin Glutamate receptor ionotropic, NMDA 2A 0 Activities

Discover Target: GRIN2A

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIN2B Tclin Glutamate receptor ionotropic, NMDA 2B 0 Activities

Discover Target: GRIN2B

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIN2C Tclin Glutamate receptor ionotropic, NMDA 2C 0 Activities

Discover Target: GRIN2C

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIN2D Tclin Glutamate receptor ionotropic, NMDA 2D 0 Activities

Discover Target: GRIN2D

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	1-methyl-16-azatetracyclo[7.6.1.0^{2,7}.0^{10,15}]hexadeca-2(7),3,5,10(15),11,13-hexaene
INCHI	InChI=1S/C16H15N/c1-16-13-8-4-2-6-11(13)10-15(17-16)12-7-3-5-9-14(12)16/h2-9,15,17H,10H2,1H3
InChi Key	LBOJYSIDWZQNJS-UHFFFAOYSA-N
Canonical SMILES	CC12NC(c3c2cccc3)Cc2c1cccc2
Isomeric SMILES	CC12C3=CC=CC=C3CC(N1)C4=CC=CC=C24
PubChem CID	1207

ChEMBL Ligand

CHEMBL442137

PubChem CID

1207

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