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STE:Homologs of yeast Sterile 7, Sterile 11, Sterile 20 kinases
IHMT-MST1-58 , CAS No.I610968, Inhibitor of serine/threonine kinase 4

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IHMT-MST1-58 , CAS No.I610968, Inhibitor of serine/threonine kinase 4

Moligand™

PubChem CID: 162477909

Item Number

I610968

Grouped product items
SKU	Size	Availability	Price	Qty
I610968-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
I610968-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,001.90

View related series

serine/threonine kinase 4 Inhibitor

Basic Description

Synonyms	compound 19
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of serine/threonine kinase 4

Associated Targets

STK3 Tchem Serine/threonine-protein kinase 3 0 Activities

Discover Target: STK3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

STK4 Tchem Serine/threonine-protein kinase 4 0 Activities

Discover Target: STK4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

NEK3 Tchem Serine/threonine-protein kinase Nek3 0 Activities

Discover Target: NEK3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	4-[[5,8-dimethyl-7-(2-methylphenyl)-6-oxo-7H-pteridin-2-yl]amino]benzenesulfonamide
INCHI	InChI=1S/C21H22N6O3S/c1-13-6-4-5-7-16(13)18-20(28)26(2)17-12-23-21(25-19(17)27(18)3)24-14-8-10-15(11-9-14)31(22,29)30/h4-12,18H,1-3H3,(H2,22,29,30)(H,23,24,25)
InChi Key	FWEIAKDAIDQPRK-UHFFFAOYSA-N
Canonical SMILES	CN1c2cnc(Nc3ccc(S(=O)(=O)N)cc3)nc2N(C)C(c2ccccc2C)C1=O
Isomeric SMILES	CC1=CC=CC=C1C2C(=O)N(C3=CN=C(N=C3N2C)NC4=CC=C(C=C4)S(=O)(=O)N)C
PubChem CID	162477909

Database links

PubChem CID	162477909

Certificates

Certificate of Analysis(COA)

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References

1. Wu Y, Qi Z, Wang B, Wang J, Liu Q, Wang A, Shi C, Zhou B, Liang Q, Wang W et al.. (2022) Discovery of IHMT-MST1-58 as a Novel, Potent, and Selective MST1 Inhibitor for the Treatment of Type 1/2 Diabetes.. J Med Chem, 129 (3): (589-97). [PMID:36037148]

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